ACS Medicinal Chemistry Letters, ISSN: 19485875
Jun Liang; Robert Blake; Jae Chang; Lori Friedman; Simon Goodacre; Steven J. Hartman; Ellen Ingalla; James Kiefer; Tracy Kleinheinz; Sharada Labadie; Jun Li; Kwong Wah Lai; Jiangpeng Liao; Vidhi Mody; Neville J. McLean; Ciara Metcalfe; Michelle Nannini; Daniel Otwine; Yingqing Ran; Nicholas C. Ray; Fabien Roussel; Amy Sambrone; Deepak Sampath; Maia Vinogradova; John Wai; Tao Wang; Kuen Yeap; Amy Young; Jason Zbieg; Birong Zhang; Xiaoping Zheng; Yu Zhong; Gina Wang
Drug Metabolism and Disposition, ISSN: 1521009X
Jae Chang; Yi-Chen Chen; Jonathan Cheong; Robert S. Jones; Jodie Pang
Molecular Pharmaceutics, ISSN: 15438392 15438384
Jae Chang; Dewakar Sangaraju; Ning Liu; Allan Jaochico; Emile Plise
Unequal absorption of radiolabeled and nonradiolabeled drug from the oral dose leads to incorrect estimates of drug absorption and circulating metabolites in a mass balance study
Drug Metabolism Letters, ISSN: 18723128
Ryan Takahashi; Jae H. Chang; Jodie Pang; Xiaorong Liang; Shuguang Ma
Unexpected equivalent potency of a constrained chromene enantiomeric pair rationalized by co-crystal structures in complex with estrogen receptor alpha
Bioorganic and Medicinal Chemistry Letters, ISSN: 0960894X
Birong Zhang; James Kiefer; Robert Blake; Jae H. Chang; Steven J. Hartman; Ellen Ingalla; Tracy Kleinheinz; Vidhi Mody; Michelle Nannini; Dan Ortwine; Yingqing Ran; Amy Sambrone; Deepak Sampath; Maia Vinogradova; Yu Zhong Yao; Jerome C. Nwachukwu; Kendall W. Nettles; Tommy Lai; Jiangpeng Liao; Xiaoping Zheng; Hai Chen; Xiaojing Wang; Jun Liang
Clinical Drug Investigation, ISSN: 11791918 11732563
Michael E. Rothenberg; Tagen; Jae H. Chang; Janel Boyce-Rustay; Michel Friesenhahn; David Hackos; Avis Hains; Dan Sutherlin; Michael Ward; William Cho
Discovery of a C-8 hydroxychromene as a potent degrader of estrogen receptor alpha with improved rat oral exposure over GDC-0927
Bioorganic and Medicinal Chemistry Letters, ISSN: 0960894X
Sharada Labadie; Jun Li; Robert Blake; Jae H. Chang; Simon Goodacre; Steven J. Hartman; Weiling Liang; James Kiefer; Tracy Kleinheinz; Tommy Lai; Jiangpeng Liao; Dan Ortwine; Vidhi Mody; Nicholas C. Ray; Fabien Roussel; Maia Vinogradova; Siew Kuen Yeap; Birong Zhang; Xiaoping Zheng; Jason Zbieg; Jun Liang; Gina Wang
Journal of Medicinal Chemistry, ISSN: 15204804 00222623
Gina Wang; Wesley P. Blackaby; Vivienne Allen; Grace Chan; Jae Chang; Po-Chang Chiang; Coura Diène; Jake Drummond; Steven Do; Eric Fan; Eric Harstad; Alastair J. Hodges; Huiyong Hu; Wei Jia; William Kofie; Aleksandr Kolesnikov; Joe Lyssikatos; Justin Ly; Mizio Matteucci; John Moffat; Veerendra Munugalavadla; Jeremy Murray; David Nash; Cameron Noland; Geoff Del Rosario; Leanne Ross; Craig Rouse; Andrew Sharpe; Dion Slaga; Minghua Sun; Vickie Tsui; Heidi Ackerly Wallweber; Shang-Fan Yu; Allen Ebens
Safety, Tolerability, and Pharmacokinetics of GDC-0276, a Novel NaV1.7 Inhibitor, in a First-in-Human, Single- and Multiple-Dose Study in Healthy Volunteers
Clinical Drug Investigation, ISSN: 11732563
Michael E. Rothenberg; Tagen; Jae H. Chang; Janel Boyce-Rustay; Michel Friesenhahn; David Hackos; Avis Hains; Dan Sutherlin; Michael Ward; William Cho
Journal of Medicinal Chemistry, ISSN: 15204804 00222623
Steven J. McKerrall; Teresa Nguyen; Kwong Wah Lai; Philippe Bergeron; Lunbin Deng; Antonio DiPasquale; Jae Chang; Jun Chen; Tania Chernov-Rogan; David Hackos; Jonathan M. Maher; Dan Ortwine; Jodie Pang; Jian Payandeh; Will Proctor; Shannon Shields; Jennifer Vogt; Pengfei Ji; Wenfeng Liu; Elisa Ballini; Lilia Schumann; Glauco Tarozzo; Girish Bankar; Sultan Chowdhury; Abid Hasan; Johnson; Kuldip Khakh; Sophia Lin; Charles J. Cohen; Christoph Dehnhardt; Brian Safina; Dan Sutherlin
Insensitivity to Pain upon Adult-Onset Deletion of Nav1.7 or Its Blockade with Selective Inhibitors
Journal of Neuroscience,
Shannon Shields; Lunbin Deng; Rebecca M. Reese; Michelle Dourado; Janet Tao; Oded Foreman; Jae H. Chang; David Hackos
Cell Reports, ISSN: 22111247
Girish Bankar; Samuel J. Goodchild; Sarah Howard; Karen Nelkenbrecher; Matthew Waldbrook; Michelle Dourado; Noah Shuart; Sophia Lin; Clint Young; Zhiwei Xie; Kuldip Khakh; Elaine Chang; Luis E. Sojo; Andrea Lindgren; Sultan Chowdhury; Shannon M. Decker; Michael Grimwood; Jean-Christophe Andrez; Christoph Dehnhardt; Jodie Pang; Jae H. Chang; Brian Safina; Dan Sutherlin; James P. Johnson; David Hackos; C. Lee Robinette; Charles J. Cohen
Journal of Medicinal Chemistry, ISSN: 15204804 00222623
Thilo Focken; Sultan Chowdhury; Alla Zenova; Michael Grimwood; Christine Chabot; Tao Sheng; Ivan Hemeon; Shannon M. Decker; Michael Wilson; Paul Bichler; Qi Jia; Shaoyi Sun; Clint Young; Sophia Lin; Samuel J. Goodchild; Noah Shuart; Elaine Chang; Zhiwei Xie; Bowen Li; Kuldip Khakh; Girish Bankar; Matthew Waldbrook; Rainbow Kwan; Karen Nelkenbrecher; Parisa Karimi Tari; Navjot Chahal; Luis E. Sojo; C. Lee Robinette; Andrew D. White; Chien-An Chen; Yi Zhang; Jodie Pang; Jae Chang; David Hackos; Johnson; Charles J. Cohen; Dan Ortwine; Dan Sutherlin; Christoph Dehnhardt; Brian Safina
Xenobiotica, ISSN: 13665928 00498254
Jae Chang; Xiaolin Zhang; Kirsten Messick; Yi-Chen Chen; Eugene Chen; Jonathan Cheong; Justin Ly
Journal of Medicinal Chemistry, ISSN: 15204804 00222623
Shaoyi Sun; Qi Jia; Alla Zenova; Michael S. Wilson; Sultan Chowdhury; Thilo Focken; Jun Li; Shannon M. Decker; Michael Grimwood; Jean-Christophe Andrez; Ivan Hemeon; Tao Sheng; Chien-An Chen; Andrew D. White; David Hackos; Lunbin Deng; Girish Bankar; Kuldip Khakh; Elaine Chang; Rainbow Kwan; Sophia Lin; Karen Nelkenbrecher; Ben Sellers; Antonio DiPasquale; Jae H. Chang; Jodie Pang; Luis E. Sojo; Andrea Lindgren; Matthew Waldbrook; Zhiwei Xie; Clint Young; James P. Johnson; C. Lee Robinette; Charles J. Cohen; Brian Safina; Dan Sutherlin; Dan Ortwine; Christoph Dehnhardt
CYP1A1-mediated intramolecular rearrangement of aminoazepane in GDC-0339
Drug Metabolism and Disposition, ISSN: 00909556
Ryan Takahashi; Gina Wang; Nathaniel Segraves; Jing Wang; Jae Chang; Cyrus Khojasteh; Shuguang Ma
Xenobiotica, ISSN: 13665928 00498254
Molly Lin; Justin Ly; Ryan Takahashi; John Chen; Alan Deese; Sarah Robinson; Aleksandr Kolesnikov; Susan Wong; Gina Wang; Jae Chang
Drug Metabolism and Disposition, ISSN: 1521009X
Ryan Takahashi; Sheerin Latham; Susan Wong; Jae Chang
Journal of Medicinal Chemistry, ISSN: 15204804
Gina Wang; Aleksandr Kolesnikov; Suzanne Brown; Grace Chan; Qi Chao; Steven Do; Jake Drummond; Allen Ebens; Ning Liu; Justin Ly; Eric Harstad; Huiyong Hu; John Moffat; Veerendra Munugalavadla; Jeremy Murray; Dion Slaga; Vickie Tsui; Matthew Volgraf; Heidi Ackerly Wallweber; Jae Chang
Journal of Pharmaceutical Sciences, ISSN: 15206017
Hsin-Fang Wu; Nadya Hristeva; Jae Chang; Xiaorong Liang; Ruina Li; Lynda A. Frassetto; Leslie Z. Benet
Drug Metabolism and Disposition, ISSN: 1521009X
Jae Chang; John Chen; Liling Liu; Kirsten Messick; Justin Ly
ACS Medicinal Chemistry Letters, ISSN: 19485875
Thilo Focken; Shifeng Liu; Navjot Chahal; Maxim Dauphinais; Michael Grimwood; Sultan Chowdhury; Ivan Hemeon; Paul Bichler; David Bogucki; Matthew Waldbrook; Girish Bankar; Luis E. Sojo; Clint Young; Sophia Lin; Noah Shuart; Rainbow Kwan; Jodie Pang; Jae Chang; Brian Safina; Dan Sutherlin; Johnson; Christoph Dehnhardt; Tarek S. Mansour; Renata M. Oballa; Charles J. Cohen; C. Lee Robinette
Bioorganic and Medicinal Chemistry Letters, ISSN: 14643405
Huiyong Hu; Gina Wang; Grace Chan; Jae Chang; Steven Do; Jake Drummond; Allen Ebens; Wendy Lee; Justin Ly; Joe Lyssikatos; Jeremy Murray; John Moffat; Qi Chao; Vickie Tsui; Heidi Ackerly Wallweber; Aleksandr Kolesnikov
ACS Medicinal Chemistry Letters, ISSN: 19485875
Gina Wang; Minghua Sun; Connie New; Spencer Nam; Wesley P. Blackaby; Alastair J. Hodges; David Nash; Mizio Matteucci; Joe Lyssikatos; Peter Fan; Suzanne Brown; Jae Chang
Drug Metabolism and Disposition, ISSN: 1521009X
Jae Chang; Justin Ly; Emile Plise; Xiaolin Zhang; Kirsten Messick; Matthew Wright; Jonathan Cheong
Molecular Pharmaceutics, ISSN: 15438384
Jae Chang; Emile Plise; Jonathan Cheong; Quynh Ho; Molly Lin
Oral Bioavailability: Basic Principles, Advanced Concepts, and Applications,
Miki Susanto Park; Jae Chang
Oral Bioavailability: Basic Principles, Advanced Concepts, and Applications,
Jae Chang; James A. Uchizono; Miki Susanto Park
Toxicological Sciences, ISSN: 10960929
Phuong Minh Nguyen; Miki Susanto Park; Marilynn Chow; Jae Chang; Lisa Wrischnik; William K. Chan