ACS Medicinal Chemistry Letters, ISSN: 19485875
Jun Liang; Robert Blake; Jae Chang; Lori Friedman; Simon Goodacre; Steven J. Hartman; Ellen Ingalla; James Kiefer; Tracy Kleinheinz; Sharada Labadie; Jun Li; Kwong Wah Lai; Jiangpeng Liao; Vidhi Mody; Neville J. McLean; Ciara Metcalfe; Michelle Nannini; Daniel Otwine; Yingqing Ran; Nicholas C. Ray; Fabien Roussel; Amy Sambrone; Deepak Sampath; Maia Vinogradova; John Wai; Tao Wang; Kuen Yeap; Amy Young; Jason Zbieg; Birong Zhang; Xiaoping Zheng; Yu Zhong; Gina Wang
Drug Metabolism and Disposition, ISSN: 1521009X 00909556
Aaron G. Bart; Ryan Takahashi; Gina Wang; Emily E. Scott
Cell, ISSN: 10974172
Jane Guan; Wei Zhou; Marc Hafner; Robert Blake; Cecile Chalouni; Irene P. Chen; Tom De Bruyn; Jennifer Giltnane; Steven J. Hartman; Amy Heidersbach; Rene Houtman; Ellen Ingalla; Kategaya; Tracy Kleinheinz; Jun Li; Scott E. Martin; Zora Modrusan; Michelle Nannini; Jason Oeh; Savita Ubhayakar; Xiaojing Wang; Ingrid Wertz; Amy Young; Mamie Yu; Deepak Sampath; Jeffrey H. Hager; Lori Friedman; Anneleen Daemen; Ciara Metcalfe
Cell Chemical Biology, ISSN: 24519448 24519456
Ingrid Wertz; Gina Wang
Organic and Biomolecular Chemistry, ISSN: 14770520
Shao-Xiong Luo; Yanzhou Liu; Michael J. Lambrecht; Dan Ortwine; Antonio DiPasquale; Jun Liang; Xiaojing Wang; Jason Zbieg; Jun Li
Discovery of a C-8 hydroxychromene as a potent degrader of estrogen receptor alpha with improved rat oral exposure over GDC-0927
Bioorganic and Medicinal Chemistry Letters, ISSN: 0960894X
Sharada Labadie; Jun Li; Robert Blake; Jae H. Chang; Simon Goodacre; Steven J. Hartman; Weiling Liang; James Kiefer; Tracy Kleinheinz; Tommy Lai; Jiangpeng Liao; Dan Ortwine; Vidhi Mody; Nicholas C. Ray; Fabien Roussel; Maia Vinogradova; Siew Kuen Yeap; Birong Zhang; Xiaoping Zheng; Jason Zbieg; Jun Liang; Gina Wang
Journal of Medicinal Chemistry, ISSN: 15204804 00222623
Gina Wang; Wesley P. Blackaby; Vivienne Allen; Grace Chan; Jae Chang; Po-Chang Chiang; Coura Diène; Jake Drummond; Steven Do; Eric Fan; Eric Harstad; Alastair J. Hodges; Huiyong Hu; Wei Jia; William Kofie; Aleksandr Kolesnikov; Joe Lyssikatos; Justin Ly; Mizio Matteucci; John Moffat; Veerendra Munugalavadla; Jeremy Murray; David Nash; Cameron Noland; Geoff Del Rosario; Leanne Ross; Craig Rouse; Andrew Sharpe; Dion Slaga; Minghua Sun; Vickie Tsui; Heidi Ackerly Wallweber; Shang-Fan Yu; Allen Ebens
Unexpected equivalent potency of a constrained chromene enantiomeric pair rationalized by co-crystal structures in complex with estrogen receptor alpha
Bioorganic and Medicinal Chemistry Letters, ISSN: 0960894X
Birong Zhang; James Kiefer; Robert Blake; Jae H. Chang; Steven J. Hartman; Ellen Ingalla; Tracy Kleinheinz; Vidhi Mody; Michelle Nannini; Dan Ortwine; Yingqing Ran; Amy Sambrone; Deepak Sampath; Maia Vinogradova; Yu Zhong Yao; Jerome C. Nwachukwu; Kendall W. Nettles; Tommy Lai; Jiangpeng Liao; Xiaoping Zheng; Hai Chen; Xiaojing Wang; Jun Liang
Nature, ISSN: 14764687 00280836
Kategaya; Paola Di Lello; Lionel Rouge; Rich Pastor; Kevin Clark; Jake Drummond; Tracy Kleinheinz; Eva Lin; John-Paul Upton; Sumit Prakash; Johanna Heideker; Mark McCleland; Maria Stella Ritorto; Dario R. Alessi; Matthias Trost; Travis Bainbridge; Michael Kwok; Taylur P. Ma; Zachary Stiffler; Bradley Brasher; Yinyan Tang; Priyadarshini Jaishankar; Brian R. Hearn; Adam R. Renslo; Michelle Arkin; Fred Cohen; Kebing Yu; Frank Peale; Florian Gnad; Matthew T. Chang; Christiaan Klijn; Beth Blackwood; Scott Martin; Bill Forrest; James Ernst; Chudi Ndubaku; Gina Wang; Maureen Beresini; Vickie Tsui; Carsten Schwerdtfeger; Robert Blake; Jeremy Murray; Till Maurer; Ingrid Wertz
CYP1A1-mediated intramolecular rearrangement of aminoazepane in GDC-0339
Drug Metabolism and Disposition, ISSN: 00909556
Ryan Takahashi; Gina Wang; Nathaniel Segraves; Jing Wang; Jae Chang; Cyrus Khojasteh; Shuguang Ma
Xenobiotica, ISSN: 13665928 00498254
Molly Lin; Justin Ly; Ryan Takahashi; John Chen; Alan Deese; Sarah Robinson; Aleksandr Kolesnikov; Susan Wong; Gina Wang; Jae Chang
ACS Medicinal Chemistry Letters, ISSN: 19485875
Gina Wang; Jim Barbosa; Peter Blomgren; Meire Bremer; Jacob Chen; James Crawford; Wei Deng; Liming Dong; Charles Eigenbrot; Steven L. Gallion; Jonathon Hau; Huiyong Hu; Adam Johnson; Arna Katewa; Jeffrey E. Kropf; Seung H. Lee; Lichuan Liu; Joe Lubach; Jen MacAluso; Patricia M. MacIejewski; Scott A. Mitchell; Dan Ortwine; Julie Dipaolo; Karin Reif; Heleen Scheerens; Aaron Schmitt; Harvey Wong; Jin-Ming Xiong; Jianjun Xu; Zhongdong Zhao; Fusheng Zhou; Kevin S. Currie; Wendy Young
Journal of Medicinal Chemistry, ISSN: 15204804
Gina Wang; Aleksandr Kolesnikov; Suzanne Brown; Grace Chan; Qi Chao; Steven Do; Jake Drummond; Allen Ebens; Ning Liu; Justin Ly; Eric Harstad; Huiyong Hu; John Moffat; Veerendra Munugalavadla; Jeremy Murray; Dion Slaga; Vickie Tsui; Matthew Volgraf; Heidi Ackerly Wallweber; Jae Chang
Bioorganic and Medicinal Chemistry Letters, ISSN: 14643405
Wendy Young; Jim Barbosa; Peter Blomgren; Meire Bremer; James Crawford; Donna Dambach; Charles Eigenbrot; Steven L. Gallion; Adam Johnson; Jeffrey E. Kropf; Seung H. Lee; Lichuan Liu; Joe Lubach; Jen MacAluso; Patricia M. MacIejewski; Scott A. Mitchell; Dan Ortwine; Julie Di Paolo; Karin Reif; Heleen Scheerens; Aaron Schmitt; Xiaojing Wang; Harvey Wong; Jin-Ming Xiong; Jianjun Xu; Christine Yu; Zhongdong Zhao; Kevin S. Currie
Bioorganic and Medicinal Chemistry Letters, ISSN: 14643405
Huiyong Hu; Gina Wang; Grace Chan; Jae Chang; Steven Do; Jake Drummond; Allen Ebens; Wendy Lee; Justin Ly; Joe Lyssikatos; Jeremy Murray; John Moffat; Qi Chao; Vickie Tsui; Heidi Ackerly Wallweber; Aleksandr Kolesnikov
ACS Medicinal Chemistry Letters, ISSN: 19485875
Gina Wang; Minghua Sun; Connie New; Spencer Nam; Wesley P. Blackaby; Alastair J. Hodges; David Nash; Mizio Matteucci; Joe Lyssikatos; Peter Fan; Suzanne Brown; Jae Chang
Bioorganic and Medicinal Chemistry Letters, ISSN: 14643405
Wendy Young; Jim Barbosa; Peter Blomgren; Meire Bremer; James Crawford; Donna Dambach; Steven L. Gallion; Sarah Hymowitz; Jeffrey E. Kropf; Seung H. Lee; Lichuan Liu; Joe Lubach; Jen MacAluso; Patricia M. MacIejewski; Brigitte Maurer; Scott A. Mitchell; Dan Ortwine; Julie Di Paolo; Karin Reif; Heleen Scheerens; Aaron Schmitt; Greg Sowell; Xiaojing Wang; Harvey Wong; Jin-Ming Xiong; Jianjun Xu; Zhongdong Zhao; Kevin S. Currie
Bioorganic and Medicinal Chemistry Letters, ISSN: 0960894X
Gina Wang; Steven Magnuson; Rich Pastor; Eric Fan; Huiyong Hu; Vickie Tsui; Wei Deng; Jeremy Murray; Micah Steffek; Heidi Ackerly Wallweber; John Moffat; Jake Drummond; Grace Chan; Eric Harstad; Allen Ebens