Unexpected equivalent potency of a constrained chromene enantiomeric pair rationalized by co-crystal structures in complex with estrogen receptor alpha
Bioorganic and Medicinal Chemistry Letters, ISSN: 0960894X
Birong Zhang; James Kiefer; Robert Blake; Jae H. Chang; Steven J. Hartman; Ellen Ingalla; Tracy Kleinheinz; Vidhi Mody; Michelle Nannini; Dan Ortwine; Yingqing Ran; Amy Sambrone; Deepak Sampath; Maia Vinogradova; Yu Zhong Yao; Jerome C. Nwachukwu; Kendall W. Nettles; Tommy Lai; Jiangpeng Liao; Xiaoping Zheng; Hai Chen; Xiaojing Wang; Jun Liang
Nature, ISSN: 14764687 00280836
Hoangdung Ho; Anh Miu; Mary Kate Alexander; Natalie K. Garcia; Angela Oh; Inna Zilberleyb; Mike Reichelt; Cary Austin; Christine Tam; Stephanie Shriver; Huiyong Hu; Sharada Labadie; Jun Liang; Lan Wang; Jian Wang; Yan Lu; Hans Purkey; John Quinn; Yvonne Franke; Kevin Clark; Maureen Beresini; Man Wah Tan; Ben Sellers; Till Maurer; Michael F. T. Koehler; Aaron Wecksler; James Kiefer; Vishal Verma; Yiming Xu; Mireille Nishiyama; Jian Payandeh; Chris Koth
ACS Medicinal Chemistry Letters, ISSN: 19485875
Terry Crawford; James E. Audia; Steve Bellon; Dan Burdick; Archana Bommi-Reddy; Alexandre Côté; Richard T Cummings; Martin Duplessis; Megan Flynn; Michael C. Hewitt; Hon-Ren Huang; Hariharan Jayaram; Ying Jiang; Shivangi Joshi; James Kiefer; Jeremy Murray; Christopher G. Nasveschuk; Adrianne Neiss; Eneida Pardo; Anthony Romero; Peter Sandy; Robert J. Sims; Yong Tang; Alexander M. Taylor; Vickie Tsui; Jian Wang; Shumei Wang; Yongyun Wang; Zhaowu Xu; Laura E. Zawadzke; Xiaoqin Zhu; Brian K Albrecht; Steven Magnuson; Andrea Cochran
Bioorganic and Medicinal Chemistry Letters, ISSN: 14643405
Terry Crawford; Steffan Vartanian; Alexandre Côté; Steve Bellon; Martin Duplessis; Megan Flynn; Michael C. Hewitt; Hon-Ren Huang; James Kiefer; Jeremy Murray; Christopher G. Nasveschuk; Eneida Pardo; Anthony Romero; Peter Sandy; Yong Tang; Alexander M. Taylor; Vickie Tsui; Jian Wang; Shumei Wang; Laura E. Zawadzke; Brian K Albrecht; Steven Magnuson; Andrea Cochran; David Stokoe
Bioorganic and Medicinal Chemistry Letters, ISSN: 14643405
Jun Liang; Sharada Labadie; Birong Zhang; Dan Ortwine; Snahel Patel; Maia Vinogradova; James Kiefer; Till Mauer; Victor S Gehling; Jean-Christophe Harmange; Richard T Cummings; Tommy Lai; Jiangpeng Liao; Xiaoping Zheng; Yichin Liu; Amy Gustafson; Erica VanderPorten; Weifeng Mao; Bianca Liederer; Gauri Deshmukh; Le An; Yingqing Ran; Marie Classon; Patrick Trojer; Peter Dragovich; Lesley Murray
Journal of Medicinal Chemistry, ISSN: 15204804
Terry Crawford; Anthony Romero; Kwong Wah Lai; Vickie Tsui; Alexander M. Taylor; Gladys Boenig; Cameron Noland; Jeremy Murray; Justin Ly; Edna Choo; Thomas Hunsaker; Emily W. Chan; Mark Merchant; Samir Kharbanda; Karen Gascoigne; Sue Kaufman; Maureen Beresini; Jiangpeng Liao; Wenfeng Liu; Kevin Chen; Zhongguo Chen; Andrew R. Conery; Alexandre Côté; Hariharan Jayaram; Ying Jiang; James Kiefer; Tracy Kleinheinz; Yingjie Li; Jonathan Maher; Eneida Pardo; Florence Poy; Kerry L. Spillane; Fei Wang; Jian Wang; Xiaocang Wei; Zhaowu Xu; Zhongya Xu; Ivana Yen; Laura E. Zawadzke; Xiaoyu Zhu; Steve Bellon; Richard T Cummings; Andrea Cochran; Brian K Albrecht; Steven Magnuson
Bioorganic and Medicinal Chemistry Letters, ISSN: 14643405
Sharada Labadie; Peter Dragovich; Richard T Cummings; Gauri Deshmukh; Amy Gustafson; Ning Han; Jean-Christophe Harmange; James Kiefer; Yue Li; Jun Liang; Bianca Liederer; Yichin Liu; Wanda Manieri; Wiefeng Mao; Lesley Murray; Dan Ortwine; Patrick Trojer; Erica VanderPorten; Maia Vinogradova; Li Wen
Bioorganic and Medicinal Chemistry Letters, ISSN: 14643405
Jun Liang; Birong Zhang; Sharada Labadie; Dan Ortwine; Maia Vinogradova; James Kiefer; Victor S Gehling; Jean-Christophe Harmange; Richard T Cummings; Tommy Lai; Jiangpeng Liao; Xiaoping Zheng; Yichin Liu; Amy Gustafson; Erica VanderPorten; Weifeng Mao; Bianca Liederer; Gauri Deshmukh; Marie Classon; Patrick Trojer; Peter Dragovich; Lesley Murray
Cytokine and Growth Factor Reviews, ISSN: 18790305
Sascha Rutz; Celine Eidenschenk; James Kiefer; Wenjun Ouyang
Nature Chemical Biology, ISSN: 15524469
Maia Vinogradova; Victor S Gehling; Amy Gustafson; Shilpi Arora; Charles Tindell; Catherine Wilson; Kaylyn E Williamson; Gulfem Guler; Pranoti Gangurde; Wanda Manieri; Jennifer Busby; Megan Flynn; Fei Lan; Hyo-jin Kim; Shobu Odate; Andrea Cochran; Yichin Liu; Matthew Wongchenko; Yibin Yang; Tommy K Cheung; Tobias Maile; Ted Lau; Mike Costa; Ganapati Hegde; Erica Jackson; Bob Pitti; David Arnott; Christopher Bailey; Steve Bellon; Richard T Cummings; Brian K Albrecht; Jean-Christophe Harmange; James Kiefer; Patrick Trojer; Marie Classon
ACS Medicinal Chemistry Letters, ISSN: 19485875
Philippe Bergeron; Michael Koehler; Beth Blackwood; Krista Bowman; Kevin Clark; Ron Firestein; James Kiefer; Klaus Maskos; Mark McCleland; Linda Orren; Sreema Ramaswamy; Laurent Salphati; Steve Schmidt; Elisabeth V. Schneider; Jiansheng Wu; Maureen Beresini
Journal of Medicinal Chemistry, ISSN: 15204804
Terry Crawford; Vickie Tsui; Megan Flynn; Shumei Wang; Alexander M. Taylor; Alexandre Côté; James E. Audia; Maureen Beresini; Dan Burdick; Richard T Cummings; Leslie A. Dakin; Martin Duplessis; Andrew C. Good; Michael C. Hewitt; Hon-Ren Huang; Hariharan Jayaram; James Kiefer; Ying Jiang; Jeremy Murray; Christopher G. Nasveschuk; Eneida Pardo; Florence Poy; Anthony Romero; Yong Tang; Jian Wang; Zhaowu Xu; Laura E. Zawadzke; Xiaoyu Zhu; Brian K Albrecht; Steven Magnuson; Steve Bellon; Andrea Cochran
ACS Medicinal Chemistry Letters, ISSN: 19485875
Alexander M. Taylor; Alexandre Côté; Michael C. Hewitt; Rich Pastor; Yves Leblanc; Christopher G. Nasveschuk; Anthony Romero; Terry Crawford; Nico Cantone; Hariharan Jayaram; Jeremy Setser; Jeremy Murray; Maureen Beresini; Gladys Boenig; Zhongguo Chen; Andrew R. Conery; Richard T Cummings; Leslie A. Dakin; Megan Flynn; Oscar Huang; Sue Kaufman; Patricia J. Keller; James Kiefer; Tommy Lai; Yingjie Li; Jiangpeng Liao; Wenfeng Liu; Henry Lu; Eneida Pardo; Vickie Tsui; Jian Wang; Yongyun Wang; Zhaowu Xu; Fen Yan; Dong Yu; Laura E. Zawadzke; Xiaoqin Zhu; Xiaoyu Zhu; Robert J. Sims; Andrea Cochran; Steve Bellon; James E. Audia; Steven Magnuson; Brian K Albrecht
ACS Medicinal Chemistry Letters, ISSN: 19485875
Michael Koehler; Philippe Bergeron; Beth Blackwood; Krista Bowman; Kevin Clark; Ron Firestein; James Kiefer; Klaus Maskos; Mark McCleland; Linda Orren; Laurent Salphati; Steve Schmidt; Elisabeth V. Schneider; Jiansheng Wu; Maureen Beresini
ACS Medicinal Chemistry Letters, ISSN: 19485875
Olivier Rene; Benjamin Fauber; Gladys Boenig; Brenda Burton; Celine Eidenschenk; Christine Everett; Alberto Gobbi; Sarah Hymowitz; Adam Johnson; James Kiefer; Marya Liimatta; Peter Lockey; Maxine Norman; Wenjun Ouyang; Heidi Ackerly Wallweber; Harvey Wong
Bioorganic and Medicinal Chemistry Letters, ISSN: 14643405
Monique B. Van Niel; Benjamin Fauber; Matthew Cartwright; Simon Gaines; Jonathan C. Killen; Olivier Rene; Stuart I. Ward; Gladys Boenig; Yuzhong Deng; Celine Eidenschenk; Christine Everett; Emanuela Gancia; Arunima Ganguli; Alberto Gobbi; Julie Hawkins; Adam Johnson; James Kiefer; Hank La; Peter Lockey; Maxine Norman; Wenjun Ouyang; Ann Qin; Nicole Wakes; Bohdan Waszkowycz; Harvey Wong
Structure, ISSN: 09692126
Jerome C. Nwachukwu; Mark R. Southern; James Kiefer; Pavel V. Afonine; Paul D. Adams; Thomas C. Terwilliger; Kendall W. Nettles
Bioorganic and Medicinal Chemistry Letters, ISSN: 0960894X
John I. Trujillo; James Kiefer; Wei Huang; Jacqueline E. Day; Joseph Moon; Gina M. Jerome; Christine P. Bono; Christine M. Kornmeier; Melanie L. Williams; Cyrille Kuhn; Glen R. Rennie; Thomas A. Wynn; Christopher P. Carron; Atli Thorarensen
Acta Crystallographica Section F: Structural Biology and Crystallization Communications, ISSN: 17443091
Troii Hall; Huey-Sheng Shieh; Jacqueline E. Day; Nicole Caspers; Jill E. Chrencik; Jennifer M. Williams; Lyle E. Pegg; Adele M. Pauley; Andrea F. Moon; Joseph M. Krahn; David H. Fischer; James Kiefer; Alfredo G. Tomasselli; Marc D. Zack