Activation of the IRE1 RNase through remodeling of the kinase front pocket by ATP-competitive ligands
Nature Communications,
Elena Ferri; Adrien Le Thomas; Heidi Ackerly Wallweber; Eric S. Day; Ben Walters; Susan Kaufman; Marie-Gabrielle Braun; Kevin Clark; Maureen Beresini; Kyle Mortara; Yung-Chia Ariel Chen; Breanna Canter; Wilson Phung; Peter Liu; Alfred Lammens; Avi Ashkenazi; Joachim Rudolph; Weiru Wang
ACS Chemical Biology, ISSN: 15548937 15548929
Dan Burdick; Nicholas Skelton; Mark Ultsch; Maureen Beresini; Charles Eigenbrot; Wei Li; Yingnan Zhang; Huy Quoc Nguyen; Monica Beltran; John Quinn; Daniel Kirchhofer
ACS Medicinal Chemistry Letters, ISSN: 19485875
Ramsay E. Beveridge; Heidi Ackerly Wallweber; Avi Ashkenazi; Maureen Beresini; Kevin R. Clark; Paul Gibbons; Elise Ghiro; Susan Kaufman; Alexandre Larivée; Melissa Leblanc; Jean-Philippe Leclerc; Alexandre Lemire; Cuong Ly; Joachim Rudolph; Jacob Schwarz; Sanjay Srivastava; Weiru Wang; Zhao; Marie-Gabrielle Braun
Disruption of IRE1α through its kinase domain attenuates multiple myeloma
Proceedings of the National Academy of Sciences of the United States of America, ISSN: 00278424
Jonathan Harnoss; Adrien Le Thomas; Anna Shemorry; Scot Marsters; David Lawrence; Min Lu; Yung-Chia Ariel Chen; Jing Qing; Klara Totpal; David Kan; Ehud Segal; Mark Merchant; Mike Reichelt; Heidi Ackerly Wallweber; Weiru Wang; Kevin Clark; Susan Kaufman; Maureen Beresini; Steven T. Laing; Wendy Sandoval; Maria Lorenzo; Jiansheng Wu; Justin Ly; Tom De Bruyn; Amy Heidersbach; Benjamin Haley; Alvin Gogineni; Robby Weimer; Dong Lee; Marie-Gabrielle Braun; Joachim Rudolph; Michael J. VanWyngarden; Daniel W. Sherbenou; Patricia Gomez-Bougie; Amiot; Diego Acosta-Alvear; Peter Walter; Avi Ashkenazi
Journal of Medicinal Chemistry, ISSN: 15204804 00222623
Shumei Wang; Vickie Tsui; Terry Crawford; James E. Audia; Dan Burdick; Maureen Beresini; Alexandre Côté; Richard T Cummings; Martin Duplessis; Megan Flynn; Michael C. Hewitt; Hon-Ren Huang; Hariharan Jayaram; Ying Jiang; Shivangi Joshi; Jeremy Murray; Christopher G. Nasveschuk; Eneida Pardo; Florence Poy; Anthony Romero; Yong Tang; Alexander M. Taylor; Jian Wang; Zhaowu Xu; Laura E. Zawadzke; Xiaoyu Zhu; Brian K Albrecht; Steven Magnuson; Steve Bellon; Andrea Cochran
Nature, ISSN: 14764687 00280836
Hoangdung Ho; Anh Miu; Mary Kate Alexander; Natalie K. Garcia; Angela Oh; Inna Zilberleyb; Mike Reichelt; Cary Austin; Christine Tam; Stephanie Shriver; Huiyong Hu; Sharada Labadie; Jun Liang; Lan Wang; Jian Wang; Yan Lu; Hans Purkey; John Quinn; Yvonne Franke; Kevin Clark; Maureen Beresini; Man Wah Tan; Ben Sellers; Till Maurer; Michael F. T. Koehler; Aaron Wecksler; James Kiefer; Vishal Verma; Yiming Xu; Mireille Nishiyama; Jian Payandeh; Chris Koth
Mechanism-specific assay design facilitates the discovery of Nav1.7-selective inhibitors
Proceedings of the National Academy of Sciences of the United States of America, ISSN: 00278424
Tania Chernov-Rogan; Tianbo Li; Gang Lu; Henry Verschoof; Kuldip Khakh; Steven W Jones; Maureen Beresini; Chang Liu; Dan Ortwine; Steven J. McKerrall; David Hackos; Dan Sutherlin; Charles J. Cohen; Jun Chen
Bioorganic and Medicinal Chemistry Letters, ISSN: 14643405 0960894X
Kwong Wah Lai; Anthony Romero; Vickie Tsui; Maureen Beresini; Gladys Boenig; Sarah M. Bronner; Kevin Chen; Zhongguo Chen; Edna Choo; Terry Crawford; Patrick Cyr; Susan Kaufman; Yingjie Li; Jiangpeng Liao; Wenfeng Liu; Justin Ly; Jeremy Murray; Weichao Shen; John Wai; Fei Wang; Caicai Zhu; Xiaoyu Zhu; Steven Magnuson
Journal of Medicinal Chemistry, ISSN: 15204804 00222623
Sarah M. Bronner; Jeremy Murray; Anthony Romero; Kwong Wah Lai; Vickie Tsui; Patrick Cyr; Maureen Beresini; Gladys Boenig; Zhongguo Chen; Edna Choo; Kevin Clark; Terry Crawford; Hariharan Jayaram; Susan Kaufman; Ruina Li; Yingjie Li; Jiangpeng Liao; Xiaorong Liang; Wenfeng Liu; Justin Ly; Jonathan M. Maher; John Wai; Fei Wang; Aijun Zheng; Xiaoyu Zhu; Steven Magnuson
Journal of Medicinal Chemistry, ISSN: 15204804 00222623
Anthony Romero; Jeremy Murray; Kwong Wah Lai; Vickie Tsui; Brian K Albrecht; Le An; Maureen Beresini; Gladys Boenig; Sarah M. Bronner; Emily Chan; Kevin Chen; Zhongguo Chen; Edna Choo; Kyle Clagg; Kevin Clark; Terry Crawford; Patrick Cyr; Denise De Almeida Nagata; Karen Gascoigne; Jane Grogan; Georgia Hatzivassiliou; Wei Huang; Thomas Hunsaker; Susan Kaufman; Stefan G. Koenig; Ruina Li; Yingjie Li; Xiaorong Liang; Jiangpeng Liao; Wenfeng Liu; Justin Ly; Jonathan M. Maher; Colin Masui; Mark Merchant; Yingqing Ran; Alexander M. Taylor; John Wai; Fei Wang; Xiaocang Wei; Dong Yu; Bing-Yan Zhu; Xiaoyu Zhu; Steven Magnuson
Nature, ISSN: 14764687 00280836
Kategaya; Paola Di Lello; Lionel Rouge; Rich Pastor; Kevin Clark; Jake Drummond; Tracy Kleinheinz; Eva Lin; John-Paul Upton; Sumit Prakash; Johanna Heideker; Mark McCleland; Maria Stella Ritorto; Dario R. Alessi; Matthias Trost; Travis Bainbridge; Michael Kwok; Taylur P. Ma; Zachary Stiffler; Bradley Brasher; Yinyan Tang; Priyadarshini Jaishankar; Brian R. Hearn; Adam R. Renslo; Michelle Arkin; Fred Cohen; Kebing Yu; Frank Peale; Florian Gnad; Matthew T. Chang; Christiaan Klijn; Beth Blackwood; Scott Martin; Bill Forrest; James Ernst; Chudi Ndubaku; Gina Wang; Maureen Beresini; Vickie Tsui; Carsten Schwerdtfeger; Robert Blake; Jeremy Murray; Till Maurer; Ingrid Wertz
Cancer Research, ISSN: 15387445 00085472
Lingyan Jin; Jesse Garcia; Emily Chan; Cecile de la Cruz; Ehud Segal; Mark Merchant; Samir Kharbanda; Ryan Raisner; Pete Haverty; Zora Modrusan; Justin Ly; Edna Choo; Sue Kaufman; Maureen Beresini; Anthony Romero; Steven Magnuson; Karen Gascoigne
Nature Structural and Molecular Biology, ISSN: 15459985 15459993
Yingnan Zhang; Mark Ultsch; Nicholas Skelton; Dan Burdick; Maureen Beresini; Wei Li Lee; Monica Beltran; Andy Peterson; John Quinn; Cecilia Chiu; Yan Wu; Steven Shia; Paul Moran; Paola Di Lello; Charles Eigenbrot; Daniel Kirchhofer
Journal of Medicinal Chemistry, ISSN: 15204804
Georgette Castanedo; Nicole Blaquiere; Maureen Beresini; Brandon Bravo; Hans Brightbill; Jacob Chen; Haifeng Cui; Charles Eigenbrot; Christine Everett; Jianwen Feng; Robert Godemann; Emily Gogol; Sarah Hymowitz; Adam Johnson; Nobuhiko Kayagaki; Pawan Bir Kohli; Kathleen Knüppel; Joachim Kraemer; Susan Krüger; Pui Loke; Paul A. McEwan; Christian A.G.N. Montalbetti; David Allen; Myron Smith; Stefan Steinbacher; Swathi Sujatha-Bhaskar; Ryan Takahashi; Xiaolu Wang; Lawren Wu; Yamin Zhang; Steven Staben
Biotechnology Progress, ISSN: 15206033
Hermann-Josef Meyer; Rebecca Turincio; Shirley Ng; Jenny Li; Blair Wilson; Pamela Chan; Mark Zak; Dorothea Reilly; Maureen Beresini; Athena Wong
Journal of Medicinal Chemistry, ISSN: 15204804
Terry Crawford; Anthony Romero; Kwong Wah Lai; Vickie Tsui; Alexander M. Taylor; Gladys Boenig; Cameron Noland; Jeremy Murray; Justin Ly; Edna Choo; Thomas Hunsaker; Emily W. Chan; Mark Merchant; Samir Kharbanda; Karen Gascoigne; Sue Kaufman; Maureen Beresini; Jiangpeng Liao; Wenfeng Liu; Kevin Chen; Zhongguo Chen; Andrew R. Conery; Alexandre Côté; Hariharan Jayaram; Ying Jiang; James Kiefer; Tracy Kleinheinz; Yingjie Li; Jonathan Maher; Eneida Pardo; Florence Poy; Kerry L. Spillane; Fei Wang; Jian Wang; Xiaocang Wei; Zhaowu Xu; Zhongya Xu; Ivana Yen; Laura E. Zawadzke; Xiaoyu Zhu; Steve Bellon; Richard T Cummings; Andrea Cochran; Brian K Albrecht; Steven Magnuson
Journal of Medicinal Chemistry, ISSN: 15204804
Terry Crawford; Vickie Tsui; Megan Flynn; Shumei Wang; Alexander M. Taylor; Alexandre Côté; James E. Audia; Maureen Beresini; Dan Burdick; Richard T Cummings; Leslie A. Dakin; Martin Duplessis; Andrew C. Good; Michael C. Hewitt; Hon-Ren Huang; Hariharan Jayaram; James Kiefer; Ying Jiang; Jeremy Murray; Christopher G. Nasveschuk; Eneida Pardo; Florence Poy; Anthony Romero; Yong Tang; Jian Wang; Zhaowu Xu; Laura E. Zawadzke; Xiaoyu Zhu; Brian K Albrecht; Steven Magnuson; Steve Bellon; Andrea Cochran
ACS Medicinal Chemistry Letters, ISSN: 19485875
Philippe Bergeron; Michael Koehler; Beth Blackwood; Krista Bowman; Kevin Clark; Ron Firestein; James Kiefer; Klaus Maskos; Mark McCleland; Linda Orren; Sreema Ramaswamy; Laurent Salphati; Steve Schmidt; Elisabeth V. Schneider; Jiansheng Wu; Maureen Beresini
ACS Medicinal Chemistry Letters, ISSN: 19485875
Alexander M. Taylor; Alexandre Côté; Michael C. Hewitt; Rich Pastor; Yves Leblanc; Christopher G. Nasveschuk; Anthony Romero; Terry Crawford; Nico Cantone; Hariharan Jayaram; Jeremy Setser; Jeremy Murray; Maureen Beresini; Gladys Boenig; Zhongguo Chen; Andrew R. Conery; Richard T Cummings; Leslie A. Dakin; Megan Flynn; Oscar Huang; Sue Kaufman; Patricia J. Keller; James Kiefer; Tommy Lai; Yingjie Li; Jiangpeng Liao; Wenfeng Liu; Henry Lu; Eneida Pardo; Vickie Tsui; Jian Wang; Yongyun Wang; Zhaowu Xu; Fen Yan; Dong Yu; Laura E. Zawadzke; Xiaoqin Zhu; Xiaoyu Zhu; Robert J. Sims; Andrea Cochran; Steve Bellon; James E. Audia; Steven Magnuson; Brian K Albrecht
ACS Medicinal Chemistry Letters, ISSN: 19485875
Michael Koehler; Philippe Bergeron; Beth Blackwood; Krista Bowman; Kevin Clark; Ron Firestein; James Kiefer; Klaus Maskos; Mark McCleland; Linda Orren; Laurent Salphati; Steve Schmidt; Elisabeth V. Schneider; Jiansheng Wu; Maureen Beresini
Journal of Laboratory Automation, ISSN: 22110690
Tim Dawes; Rebecca Turincio; Steven Jones; Richie Rodriguez; Dhireshan Gadiagellan; Peter Thana; Kevin Clark; Amy Gustafson; Linda Orren; Marya Liimatta; Daniel Gross; Till Maurer; Maureen Beresini
Journal of Biomolecular Screening, ISSN: 1552454X
Maureen Beresini; Yichin Liu; Tim Dawes; Kevin Clark; Linda Orren; Steve Schmidt; Rebecca Turincio; Steven Jones; Richie Rodriguez; Peter Thana; Dan Hascall; Daniel Gross; Nicholas Skelton
European Journal of Medicinal Chemistry, ISSN: 02235234
Jun Liang; Vickie Tsui; Anne Van Abbema; Liang Bao; Kathy Barrett; Maureen Beresini; Leo Berezhkovskiy; Wade Blair; Christine Chang; James Driscoll; Charles Eigenbrot; Nico Ghilardi; Paul Gibbons; Jason Halladay; Adam Johnson; Pawan Bir Kohli; Yingjie Lai; Marya Liimatta; Priscilla Mantik; Kapil Menghrajani; Jeremy Murray; Amy Sambrone; Yisong Xiao; Steven Shia; Young Shin; Jan Smith; Sue Sohn; Mark Stanley; Mark Ultsch; Birong Zhang; Lawren Wu; Steven Magnuson
Journal of Medicinal Chemistry, ISSN: 00222623
John Flygare; Maureen Beresini; Nageshwar Budha; Helen Chan; Iris Chan; Sravanthi Cheeti; Fred Cohen; Kurt Deshayes; Karl Doerner; Gail Eckhardt; Linda Orren; Bainian Feng; Matthew C. Franklin; Stacy Reisner; Lewis Gazzard; Jason Halladay; Sarah Hymowitz; Hank La; Patricia M. LoRusso; Brigitte Maurer; Lesley Murray; Emile Plise; Clifford Quan; Daniel Stephan; Young Shin; Jeffrey Tom; Vickie Tsui; Joann M. Um; Eugene Varfolomeev; Domagoj Vucic; Andrew Wagner; Heidi Ackerly Wallweber; Lan Wang; Joseph Ware; Kobe Wen; Harvey Wong; Jonathan Wong; Melisa Wong; Susan Wong; Ron Yu; Kerry Zobel; Wayne Fairbrother
Journal of Biomolecular Screening, ISSN: 10870571
Yichin Liu; Maureen Beresini; Adam Johnson; Bob Mintzer; Kinjal Shah; Kevin Clark; Steve Schmidt; Cris Lewis; Marya Liimatta; Linda Orren; Amy Gustafson; Chris Heise
Journal of Immunological Methods, ISSN: 00221759
Yanmei Lu; Jean-Michel Vernes; Nancy Chiang; Qinglin Ou; Jiabing Ding; Camellia Adams; Kyu Hong; Bao-Tran Truong; Domingos Ng; Amy Shen; Gerry Nakamura; Qian Gong; Leonard G. Presta; Maureen Beresini; Bob Kelley; Henry Lowman; Wai Lee Wong; Gloria Meng
Protein Science, ISSN: 09618368
Susan Keating; Kevin Clark; Lisa D. Stefanich; Fred Arellano; Caroline Phelps Edwards; Sarah C. Bodary; Steven A. Spencer; Thomas R. Gadek; James Marsters; Maureen Beresini
Journal of Biological Chemistry, ISSN: 00219258
Alan Olivero; Charles Eigenbrot; Rich Goldsmith; Kirk Robarge; Dean R. Artis; John Flygare; Thomas Rawson; Dan Sutherlin; Saloumeh Kadkhodayan; Maureen Beresini; Linda Orren; Geralyn G. Deguzman; David W. Banner; Mark Ultsch; Ulla Marzec; Stephen R. Hanson; Ken Refino; Stuart Bunting; Daniel Kirchhofer
Bioorganic and Medicinal Chemistry Letters, ISSN: 0960894X
Dan Burdick; James Marsters; Ignacio Aliagas; Mark Stanley; Maureen Beresini; Kevin Clark; Robert S. McDowell; Thomas R. Gadek
Bioorganic and Medicinal Chemistry Letters, ISSN: 0960894X
Kerry Zobel; Michael Koehler; Maureen Beresini; Lisa D. Caris; Daniel Combs
Bioorganic and Medicinal Chemistry Letters, ISSN: 0960894X
Dan Burdick; Ken Paris; Kenneth Weese; Mark Stanley; Maureen Beresini; Kevin Clark; Robert S. McDowell; James Marsters; Thomas R. Gadek
Bioorganic and Medicinal Chemistry Letters, ISSN: 0960894X
Michael Koehler; Kerry Zobel; Maureen Beresini; Lisa D. Caris; Daniel Combs; Brian Paasch; Bob Lazarus
Bioorganic and Medicinal Chemistry Letters, ISSN: 0960894X
Georgette Castanedo; Fredrick C. Sailes; Dubree; John Nicholas; Lisa D. Caris; Kevin Clark; Susan Keating; Maureen Beresini; Henry Chiu; Sherman Fong; James Marsters; David Jackson; Dan Sutherlin
Osteoarthritis and Cartilage, ISSN: 10634584
Liping Cai; Franklin W. Okumu; Jeffrey L. Cleland; Maureen Beresini; Deborah Hogue; Zhonghua Lin; Ellen Filvaroff
Journal of Medicinal Chemistry, ISSN: 00222623
Dubree; Dean R. Artis; Georgette Castanedo; James Marsters; Dan Sutherlin; Lisa D. Caris; Kevin Clark; Susan Keating; Maureen Beresini; Henry Chiu; Sherman Fong; Henry Lowman; Nicholas Skelton; David Jackson
Journal of Biological Chemistry, ISSN: 00219258
Camenisch; Maria T. Pisabarro; Dan Sherman; Joe Kowalski; Mark Nagel; Phil Hass; Ming-Hong Xie; Austin L. Gurney; Sarah C. Bodary; Xiao-Huan Liang; Kevin Clark; Maureen Beresini; Napoleone Ferrara; Hans-Peter Gerber
Science, ISSN: 00368075
Thomas R. Gadek; Dan Burdick; Robert S. McDowell; Mark Stanley; James Marsters; Ken Paris; David Arthur Oare; Mark Reynolds; Carmen Ladner; Kimberly Zioncheck; Wyne Lee; Peter Gribling; Mark Dennis; Nicholas Skelton; Daniel B. Tumas; Kevin Clark; Susan Keating; Maureen Beresini; Jefferson W Tilley; Leonard G. Presta; Sarah C. Bodary
Proceedings of SPIE - The International Society for Optical Engineering, ISSN: 0277786X
Susan Keating; James Marsters; Maureen Beresini; Carmen Ladner; Kimberly Zioncheck; Kevin Clark; Fred Arellano; Sarah C. Bodary
Biopolymers - Peptide Science Section, ISSN: 00063525
Clifford Quan; Nicholas Skelton; Kevin Clark; David Jackson; Mark Renz; Henry Chiu; Susan Keating; Maureen Beresini; Sherman Fong; Dean R. Artis
Journal of the American Chemical Society, ISSN: 00027863
Charles Y. Cho; R. Scott Youngquist; Sari J. Paikoff; Maureen Beresini; Andrea R. Hebert; Lea Berleau; Corey W. Liu; David E. Wemmer; Thomas Keough; Peter G. Schultz
Thrombosis and Haemostasis, ISSN: 03406245
Ken Refino; Nishit Bachulal Modi; Sherry Bullens; Cheryl Pater; Terry Lipari; Kirk Robarge; Brent Blackburn; Maureen Beresini; Thomas Weller; Beat Steiner; Stuart Bunting
Journal of Medicinal Chemistry, ISSN: 00222623
Thomas Weller; Leo Alig; Maureen Beresini; Brent Blackburn; Stuart Bunting; Paul Hadváry; Marianne Hürzeler Müller; Dietmar Knopp; Bernard Levet-Trafit; Terry Lipari; Nishit Bachulal Modi; Marcel Müller; Ken Refino; Monique Schmitt; Peter Schönholzer; Sabine Weiss; Beat Steiner
Biochemical and Biophysical Research Communications, ISSN: 0006291X
Amit Kumar; Maureen Beresini; Punita Dhawan; Kamal D. Mehta
Electrophoresis, ISSN: 15222683
Maureen Beresini; Sugarman; Shepard; Lois B. Epstein