Preclinical Safety Assessment of a Highly Selective and Potent Dual Small-Molecule Inhibitor of CBP/P300 in Rats and Dogs
Toxicologic Pathology, ISSN: 01926233
Paula Katavolos; Cain; Cindy A. Farman; Anthony Romero; Steven Magnuson; Justin Ly; Edna Choo; Anand Kumar Katakam; Roxanne Andaya; Jonathan M. Maher
A Non-covalent Ligand Reveals Biased Agonism of the TRPA1 Ion Channel
Neuron, ISSN: 08966273
Chang Liu; Rebecca M. Reese; Simon Vu; Lionel Rouge; Shannon Shields; Satoko Kakiuchi-Kiyota; Huifen Chen; Kevin Johnson; Yu Patrick Shi; Tania Chernov-Rogan; Demi Maria Zabala Greiner; Pawan Bir Kohli; David Hackos; Bobby Brillantes; Christine Tam; Tianbo Li; Jianyong Wang; Brian Safina; Steven Magnuson; Matthew Volgraf; Jian Payandeh; Jie Zheng; Alexis Rohou; Jun Chen
Proceedings of the National Academy of Sciences of the United States of America, ISSN: 10916490 00278424
Tania Chernov-Rogan; Eleonora Gianti; Chang Liu; Elisia Villemure; Andrew P. Cridland; Xiaoyu Hu; Elisa Ballini; Wienke Lange; Heike Deisemann; Tianbo Li; Stuart I. Ward; David Hackos; Steven Magnuson; Brian Safina; Michael L. Klein; Matthew Volgraf; Vincenzo Carnevale; Jun Chen
CBP/p300 drives the differentiation of regulatory T cells through transcriptional and non-transcriptional mechanisms
Cancer Research, ISSN: 00085472
Joseph Castillo; Esther Wu; Christopher Lowe; Shrividhya Srinivasan; Mccord; Marie-Claire Wagle; Sangeeta Jayakar; Melissa Gonzalez Edick; Jeff Eastham; Bonnie Liu; Katherine E. Hutchinson; Wendell Jones; Matthew P. Stokes; Somayeh S. Tarighat; Tom Holcomb; Andrew Glibicky; Anthony Romero; Steven Magnuson; Shih-Min A. Huang; Vicki Plaks; Jennifer Giltnane; Mark Lackner; Zineb Mounir
Cell Reports, ISSN: 22111247
Denise De Almeida Nagata; Eugene Chiang; Suchit Jhunjhunwala; Patrick Caplazi; Vidhyalakshmi Arumugam; Zora Modrusan; Emily Chan; Mark Merchant; Lingyan Jin; David Arnott; Anthony Romero; Steven Magnuson; Karen Gascoigne; Jane Grogan
Journal of Medicinal Chemistry, ISSN: 15204804 00222623
Shumei Wang; Vickie Tsui; Terry Crawford; James E. Audia; Dan Burdick; Maureen Beresini; Alexandre Côté; Richard T Cummings; Martin Duplessis; Megan Flynn; Michael C. Hewitt; Hon-Ren Huang; Hariharan Jayaram; Ying Jiang; Shivangi Joshi; Jeremy Murray; Christopher G. Nasveschuk; Eneida Pardo; Florence Poy; Anthony Romero; Yong Tang; Alexander M. Taylor; Jian Wang; Zhaowu Xu; Laura E. Zawadzke; Xiaoyu Zhu; Brian K Albrecht; Steven Magnuson; Steve Bellon; Andrea Cochran
Cell Reports, ISSN: 22111247
Ryan Raisner; Samir Kharbanda; Lingyan Jin; Edwin Jeng; Emily Chan; Mark Merchant; Matthias Peter; Russell Bainer; Tommy K Cheung; David Arnott; Megan Flynn; Anthony Romero; Steven Magnuson; Karen Gascoigne
Bioorganic and Medicinal Chemistry Letters, ISSN: 14643405 0960894X
Kwong Wah Lai; Anthony Romero; Vickie Tsui; Maureen Beresini; Gladys Boenig; Sarah M. Bronner; Kevin Chen; Zhongguo Chen; Edna Choo; Terry Crawford; Patrick Cyr; Susan Kaufman; Yingjie Li; Jiangpeng Liao; Wenfeng Liu; Justin Ly; Jeremy Murray; Weichao Shen; John Wai; Fei Wang; Caicai Zhu; Xiaoyu Zhu; Steven Magnuson
Journal of Medicinal Chemistry, ISSN: 15204804 00222623
Sarah M. Bronner; Jeremy Murray; Anthony Romero; Kwong Wah Lai; Vickie Tsui; Patrick Cyr; Maureen Beresini; Gladys Boenig; Zhongguo Chen; Edna Choo; Kevin Clark; Terry Crawford; Hariharan Jayaram; Susan Kaufman; Ruina Li; Yingjie Li; Jiangpeng Liao; Xiaorong Liang; Wenfeng Liu; Justin Ly; Jonathan M. Maher; John Wai; Fei Wang; Aijun Zheng; Xiaoyu Zhu; Steven Magnuson
Journal of Medicinal Chemistry, ISSN: 15204804 00222623
Anthony Romero; Jeremy Murray; Kwong Wah Lai; Vickie Tsui; Brian K Albrecht; Le An; Maureen Beresini; Gladys Boenig; Sarah M. Bronner; Emily Chan; Kevin Chen; Zhongguo Chen; Edna Choo; Kyle Clagg; Kevin Clark; Terry Crawford; Patrick Cyr; Denise De Almeida Nagata; Karen Gascoigne; Jane Grogan; Georgia Hatzivassiliou; Wei Huang; Thomas Hunsaker; Susan Kaufman; Stefan G. Koenig; Ruina Li; Yingjie Li; Xiaorong Liang; Jiangpeng Liao; Wenfeng Liu; Justin Ly; Jonathan M. Maher; Colin Masui; Mark Merchant; Yingqing Ran; Alexander M. Taylor; John Wai; Fei Wang; Xiaocang Wei; Dong Yu; Bing-Yan Zhu; Xiaoyu Zhu; Steven Magnuson
Cancer Research, ISSN: 15387445 00085472
Lingyan Jin; Jesse Garcia; Emily Chan; Cecile de la Cruz; Ehud Segal; Mark Merchant; Samir Kharbanda; Ryan Raisner; Pete Haverty; Zora Modrusan; Justin Ly; Edna Choo; Sue Kaufman; Maureen Beresini; Anthony Romero; Steven Magnuson; Karen Gascoigne
ACS Medicinal Chemistry Letters, ISSN: 19485875
Terry Crawford; James E. Audia; Steve Bellon; Dan Burdick; Archana Bommi-Reddy; Alexandre Côté; Richard T Cummings; Martin Duplessis; Megan Flynn; Michael C. Hewitt; Hon-Ren Huang; Hariharan Jayaram; Ying Jiang; Shivangi Joshi; James Kiefer; Jeremy Murray; Christopher G. Nasveschuk; Adrianne Neiss; Eneida Pardo; Anthony Romero; Peter Sandy; Robert J. Sims; Yong Tang; Alexander M. Taylor; Vickie Tsui; Jian Wang; Shumei Wang; Yongyun Wang; Zhaowu Xu; Laura E. Zawadzke; Xiaoqin Zhu; Brian K Albrecht; Steven Magnuson; Andrea Cochran
Bioorganic and Medicinal Chemistry Letters, ISSN: 14643405
Terry Crawford; Steffan Vartanian; Alexandre Côté; Steve Bellon; Martin Duplessis; Megan Flynn; Michael C. Hewitt; Hon-Ren Huang; James Kiefer; Jeremy Murray; Christopher G. Nasveschuk; Eneida Pardo; Anthony Romero; Peter Sandy; Yong Tang; Alexander M. Taylor; Vickie Tsui; Jian Wang; Shumei Wang; Laura E. Zawadzke; Brian K Albrecht; Steven Magnuson; Andrea Cochran; David Stokoe
Bioorganic and Medicinal Chemistry Letters, ISSN: 14643405 0960894X
Jun Liang; Anne Van Abbema; Mercedesz Balazs; Kathy Barrett; Leo Berezhkovsky; Wade Blair; Christine Chang; Donnie Delarosa; Jason DeVoss; James Driscoll; Charles Eigenbrot; Simon Goodacre; Nico Ghilardi; Calum Macleod; Adam Johnson; Pawan Bir Kohli; Yingjie Lai; Zhonghua Lin; Priscilla Mantik; Kapil Menghrajani; Hieu Nguyen; Ivan Peng; Amy Sambrone; Steven Shia; Jan Smith; Sue Sohn; Vickie Tsui; Mark Ultsch; Karen Williams; Lawren Wu; Wenqian Yang; Birong Zhang; Steven Magnuson
Journal of Medicinal Chemistry, ISSN: 15204804
Terry Crawford; Anthony Romero; Kwong Wah Lai; Vickie Tsui; Alexander M. Taylor; Gladys Boenig; Cameron Noland; Jeremy Murray; Justin Ly; Edna Choo; Thomas Hunsaker; Emily W. Chan; Mark Merchant; Samir Kharbanda; Karen Gascoigne; Sue Kaufman; Maureen Beresini; Jiangpeng Liao; Wenfeng Liu; Kevin Chen; Zhongguo Chen; Andrew R. Conery; Alexandre Côté; Hariharan Jayaram; Ying Jiang; James Kiefer; Tracy Kleinheinz; Yingjie Li; Jonathan Maher; Eneida Pardo; Florence Poy; Kerry L. Spillane; Fei Wang; Jian Wang; Xiaocang Wei; Zhaowu Xu; Zhongya Xu; Ivana Yen; Laura E. Zawadzke; Xiaoyu Zhu; Steve Bellon; Richard T Cummings; Andrea Cochran; Brian K Albrecht; Steven Magnuson
Journal of Biological Chemistry, ISSN: 1083351X
Srimoyee Ghosh; Alexander M. Taylor; Melissa Chin; Hon-Ren Huang; Andrew R. Conery; Jennifer A. Mertz; Andres Salmeron; Pranal J. Dakle; Deanna Mele; Alexandre Côté; Hari Jayaram; Jeremy Setser; Florence Poy; Georgia Hatzivassiliou; Denise de Almeida Nagata; Peter Sandy; Charlie Hatton; Anthony Romero; Eugene Chiang; Thornik Reimer; Terry Crawford; Eneida Pardo; Venita G. Watson; Vickie Tsui; Andrea Cochran; Laura E. Zawadzke; Jean-Christophe Harmange; James E. Audia; Barbara M. Bryant; Richard T Cummings; Steven Magnuson; Jane Grogan; Steve Bellon; Brian K Albrecht; Robert J. Sims; Jose M. Lora
Journal of Medicinal Chemistry, ISSN: 15204804
Terry Crawford; Vickie Tsui; Megan Flynn; Shumei Wang; Alexander M. Taylor; Alexandre Côté; James E. Audia; Maureen Beresini; Dan Burdick; Richard T Cummings; Leslie A. Dakin; Martin Duplessis; Andrew C. Good; Michael C. Hewitt; Hon-Ren Huang; Hariharan Jayaram; James Kiefer; Ying Jiang; Jeremy Murray; Christopher G. Nasveschuk; Eneida Pardo; Florence Poy; Anthony Romero; Yong Tang; Jian Wang; Zhaowu Xu; Laura E. Zawadzke; Xiaoyu Zhu; Brian K Albrecht; Steven Magnuson; Steve Bellon; Andrea Cochran
ACS Medicinal Chemistry Letters, ISSN: 19485875
Alexander M. Taylor; Alexandre Côté; Michael C. Hewitt; Rich Pastor; Yves Leblanc; Christopher G. Nasveschuk; Anthony Romero; Terry Crawford; Nico Cantone; Hariharan Jayaram; Jeremy Setser; Jeremy Murray; Maureen Beresini; Gladys Boenig; Zhongguo Chen; Andrew R. Conery; Richard T Cummings; Leslie A. Dakin; Megan Flynn; Oscar Huang; Sue Kaufman; Patricia J. Keller; James Kiefer; Tommy Lai; Yingjie Li; Jiangpeng Liao; Wenfeng Liu; Henry Lu; Eneida Pardo; Vickie Tsui; Jian Wang; Yongyun Wang; Zhaowu Xu; Fen Yan; Dong Yu; Laura E. Zawadzke; Xiaoqin Zhu; Xiaoyu Zhu; Robert J. Sims; Andrea Cochran; Steve Bellon; James E. Audia; Steven Magnuson; Brian K Albrecht
Cancer Research, ISSN: 15387445
John P. McGrath; Kaylyn E Williamson; Srividya Balasubramanian; Shobu Odate; Shilpi Arora; Charlie Hatton; Thomas M. Edwards; Thomas O'Brien; Steven Magnuson; David Stokoe; Danette L. Daniels; Barbara M. Bryant; Patrick Trojer
Journal of Medicinal Chemistry, ISSN: 15204804
Anthony Romero; Alexander M. Taylor; Terry Crawford; Vickie Tsui; Alexandre Côté; Steven Magnuson
Bioorganic and Medicinal Chemistry Letters, ISSN: 14643405
Dan Burdick; Shumei Wang; Chris Heise; Borlan Pan; Jake Drummond; Peter Yin; Lauren Goeser; Steven Magnuson; Jeff Blaney; John Moffat; Weiru Wang; Huifen Chen
Journal of Medicinal Chemistry, ISSN: 15204804
Giovanni Cervi; Paola Magnaghi; Daniela Asa; Nilla Avanzi; Alessandra Badari; Daniela Borghi; Michele Caruso; Alessandra Cirla; Liviana Cozzi; Eduard Felder; Arturo Galvani; Fabio Gasparri; Antonio Lomolino; Steven Magnuson; Beatrice Malgesini; Ilaria Motto; Maurizio Pasi; Simona Rizzi; Barbara Salom; Graziella Sorrentino; Sonia Troiani; Barbara Valsasina; Thomas O'Brien; Antonella Isacchi; Daniele Donati; Roberto D'Alessio
Bioorganic and Medicinal Chemistry Letters, ISSN: 14643405
Lan Wang; Mark Stanley; Jason Boggs; Terry Crawford; Brandon Bravo; Tony Giannetti; Seth Harris; Steven Magnuson; Jim Nonomiya; Steve Schmidt; Ping Wu; Weilan Ye; Stephen Gould; Lesley Murray; Chudi Ndubaku; Huifen Chen
Bioorganic and Medicinal Chemistry Letters, ISSN: 14643405
Rich Pastor; Jason Burch; Steven Magnuson; Dan Ortwine; Yuan Chen; Michael De La Torre; Xiao Ding; Charles Eigenbrot; Adam Johnson; Marya Liimatta; Yichin Liu; Steven Shia; Xiaolu Wang; Lawren Wu; Zhonghua Pei
Journal of Medicinal Chemistry, ISSN: 15204804
Terry Crawford; Chudi Ndubaku; Huifen Chen; Jason Boggs; Brandon Bravo; Kelly Delatorre; Tony Giannetti; Stephen Gould; Seth Harris; Steven Magnuson; Erin McNamara; Lesley Murray; Jim Nonomiya; Amy Sambrone; Steve Schmidt; Tanya Smyczek; Mark Stanley; Philip Vitorino; Lan Wang; Kristina West; Ping Wu; Weilan Ye
Journal of Medicinal Chemistry, ISSN: 15204804
Benjamin Fauber; Steven Magnuson
Journal of Heterocyclic Chemistry, ISSN: 19435193
Jun Liang; Valerie Dorman Soucy; Vickie Tusi; Yanzhou Liu; Birong Zhang; Yingjie Lai; Steven Magnuson; Bing-Yan Zhu; Fangdao Wang; Jinghao Gu; Qingfen Zhang; Yuan Wu; Wei Deng; Wenqian Yang
Bioorganic and Medicinal Chemistry Letters, ISSN: 0960894X
Mike Siu; Rich Pastor; Wendy Liu; Kathy Barrett; Megan Berry Swadell; Wade Blair; Christine Chang; Jacob Chen; Charles Eigenbrot; Nico Ghilardi; Paul Gibbons; Haiying He; Christopher A. Hurley; Jane Kenny; Cyrus Khojasteh; Hoa Le; Leslie Lee; Joe Lyssikatos; Steven Magnuson; Rebecca Pulk; Vickie Tsui; Mark Ultsch; Yisong Xiao; Bing-Yan Zhu; Deepak Sampath
Journal of Immunology, ISSN: 00221767
Sue Sohn; Kathy Barrett; Anne Van Abbema; Christine Chang; Pawan Bir Kohli; Hidenobu Kanda; Janice Smith; Yingjie Lai; Aihe Zhou; Birong Zhang; Wenqian Yang; Karen Williams; Calum Macleod; Christopher A. Hurley; Janusz J. Kulagowski; Nicholas Lewin-Koh; Hart S. Dengler; Adam Johnson; Nico Ghilardi; Mark Zak; Jun Liang; Wade Blair; Steven Magnuson; Lawren Wu
European Journal of Medicinal Chemistry, ISSN: 02235234
Jun Liang; Vickie Tsui; Anne Van Abbema; Liang Bao; Kathy Barrett; Maureen Beresini; Leo Berezhkovskiy; Wade Blair; Christine Chang; James Driscoll; Charles Eigenbrot; Nico Ghilardi; Paul Gibbons; Jason Halladay; Adam Johnson; Pawan Bir Kohli; Yingjie Lai; Marya Liimatta; Priscilla Mantik; Kapil Menghrajani; Jeremy Murray; Amy Sambrone; Yisong Xiao; Steven Shia; Young Shin; Jan Smith; Sue Sohn; Mark Stanley; Mark Ultsch; Birong Zhang; Lawren Wu; Steven Magnuson
Journal of Medicinal Chemistry, ISSN: 00222623
Jun Liang; Anne Van Abbema; Mercedesz Balazs; Kathy Barrett; Leo Berezhkovsky; Wade Blair; Christine Chang; Donnie Delarosa; Jason DeVoss; James Driscoll; Charles Eigenbrot; Nico Ghilardi; Paul Gibbons; Jason Halladay; Adam Johnson; Pawan Bir Kohli; Yingjie Lai; Yanzhou Liu; Joe Lyssikatos; Priscilla Mantik; Kapil Menghrajani; Jeremy Murray; Ivan Peng; Amy Sambrone; Steven Shia; Young Shin; Jan Smith; Sue Sohn; Vickie Tsui; Mark Ultsch; Lawren Wu; Yisong Xiao; Wenqian Yang; Judy Young; Birong Zhang; Bing-Yan Zhu; Steven Magnuson
Bioorganic and Medicinal Chemistry Letters, ISSN: 0960894X
Gina Wang; Steven Magnuson; Rich Pastor; Eric Fan; Huiyong Hu; Vickie Tsui; Wei Deng; Jeremy Murray; Micah Steffek; Heidi Ackerly Wallweber; John Moffat; Jake Drummond; Grace Chan; Eric Harstad; Allen Ebens
Cancer Research, ISSN: 00085472
Ted Lau; Emily Chan; Marinella Callow; Jo Waaler; Jason Boggs; Robert A. Blake; Steven Magnuson; Amy Sambrone; Melissa Schutten; Ron Firestein; Ondrej Machon; Vladimir Korinek; Edna Choo; Dolo Diaz; Mark Merchant; Paul Polakis; Daniel D. Holsworth; Stefan Krauss; Mike Costa
Tetrahedron Letters, ISSN: 00404039
Olivier Rene; Alexandra Souverneva; Steven Magnuson; Benjamin Fauber
Journal of Medicinal Chemistry, ISSN: 15204804
Paolo Polucci; Paola Magnaghi; Mauro Angiolini; Daniela Asa; Nilla Avanzi; Alessandra Badari; Jay Bertrand; Elena Casale; Silvia Cauteruccio; Alessandra Cirla; Liviana Cozzi; Arturo Galvani; Peter Jackson; Yichin Liu; Steven Magnuson; Beatrice Malgesini; Stefano Nuvoloni; Christian Orrenius; Federico Riccardi Sirtori; Laura Riceputi; Simona Rizzi; Beatrice Trucchi; Thomas O'Brien; Antonella Isacchi; Daniele Donati; Roberto D'Alessio
Journal of Medicinal Chemistry, ISSN: 00222623
Emily Hanan; Anne Van Abbema; Kathy Barrett; Wade Blair; Jeff Blaney; Christine Chang; Charles Eigenbrot; Sean Flynn; Paul Gibbons; Christopher A. Hurley; Jane Kenny; Janusz J. Kulagowski; Leslie Lee; Steven Magnuson; Claire Morris; Jeremy Murray; Rich Pastor; Thomas Rawson; Mike Siu; Mark Ultsch; Aihe Zhou; Deepak Sampath; Joe Lyssikatos
Proteins: Structure, Function and Bioinformatics, ISSN: 08873585
Vickie Tsui; Paul Gibbons; Mark Ultsch; Kyle Mortara; Christine Chang; Wade Blair; Rebecca Pulk; Mark Stanley; Melissa Starovasnik; David Williams; Maria Lamers; Phillip Leonard; Steven Magnuson; Jun Liang; Charles Eigenbrot