Drug Metabolism and Disposition, ISSN: 1521009X
Xingrong Liu; Xiaorong Liang; Jenninfer LeCouter; Savita Ubhayakar; Jacob Chen; Jay Cheng; Tom Lee; Joe Lubach; Jim Nonomiya; Sheerin Latham; Cristine Quiason-Huynh; Eric G. Solon; Matthew Wright; Marcel Hop; Tim Heffron
Hematopoietic Progenitor Kinase-1 Structure in a Domain-Swapped Dimer
Structure,
Ping Wu; Christopher J. Sneeringer; Keith E. Pitts; Eric S. Day; Bryan Chan; Binqing Wei; Isabelle Lehoux; Kyle Mortara; Hong Li; Jiansheng Wu; Yvonne Franke; John Moffat; Jane Grogan; Tim Heffron; Weiru Wang
Design of a brain-penetrant CDK4/6 inhibitor for glioblastoma
Bioorganic and Medicinal Chemistry Letters, ISSN: 0960894X
Sarah M. Bronner; Karl A. Merrick; Jeremy Murray; Laurent Salphati; John Moffat; Jodie Pang; Christopher Sneeringer; Nick Dompe; Patrick Cyr; Hans Purkey; Gladys de Leon Boenig; Jun Li; Aleksandr Kolesnikov; Larouche-Gauthier; Kwong Wah Lai; Xiaoli Shen; Samuel Aubert-Nicol; Yi-Chen Chen; Jonathan Cheong; James Crawford; Marc Hafner; Pouyan Haghshenas; Araz Jakalian; Jean-Philippe Leclerc; Ngiap-Kie Lim; Thomas O'Brien; Emile Plise; Shalan; Claudio Sturino; John Wai; Yang Xiao; Peter Yin; Zhao; Stephen Gould; Alan Olivero; Tim Heffron
ACS Symposium Series, ISSN: 19475918 00976156
Remy Angelaud; Steven Staben; Tim Heffron; Andreas M. Schuster; Frederic St-Jean
Neuro-Oncology, ISSN: 15235866 15228517
Tim Heffron
Drug Metabolism and Disposition, ISSN: 1521009X
Laurent Salphati; Bruno Alicke; Tim Heffron; Sheerin Latham; Merry Nishimura; Cao; Rick Carano; Jonathan Cheong; Joan Greve; Hartmut Koeppen; Shari Lau; Leslie Lee; Michelle Nannini; Jodie Pang; Emile Plise; Cristine Quiason; Linda Rangell; Xiaolin Zhang; Stephen Gould; Heidi Phillips; Alan Olivero
Journal of Medicinal Chemistry, ISSN: 15204804
Bryan Chan; Emily Hanan; Krista Bowman; Callie Bryan; Dan Burdick; Emily Chan; Yuan Chen; Saundra Clausen; Trisha Dela Vega; Jenna Dotson; Charles Eigenbrot; Richard Elliott; Robert Heald; Philip Jackson; Jamie D. Knight; Hank La; Michael Lainchbury; Shiva Malek; Hans Purkey; Gabriele Schaefer; Steve Schmidt; Eileen M. Seward; Steve Sideris; Lily Shao; Shumei Wang; Siew Kuen Yeap; Ivana Yen; Christine Yu; Tim Heffron
ACS Medicinal Chemistry Letters, ISSN: 19485875
Tim Heffron; Chudi Ndubaku; Laurent Salphati; Bruno Alicke; Jonathan Cheong; Joy Drobnick; Kyle Edgar; Stephen Gould; Leslie Lee; John Lesnick; Cris Lewis; Jim Nonomiya; Jodie Pang; Emile Plise; Steve Sideris; Jeffrey Wallin; Lan Wang; Xiaolin Zhang; Alan Olivero
Journal of Medicinal Chemistry, ISSN: 15204804
Tim Heffron; Robert Heald; Chudi Ndubaku; Binqing Wei; Martin Augistin; Steven Do; Kyle Edgar; Charles Eigenbrot; Lori Friedman; Emanuela Gancia; Philip Jackson; Graham Jones; Aleksandr Kolesnikov; Leslie B. Lee; John Lesnick; Cris Lewis; Neville J. McLean; Mario Mörtl; Jim Nonomiya; Jodie Pang; Steve Price; Wei Wei Prior; Laurent Salphati; Steve Sideris; Steven Staben; Stefan Steinbacher; Vickie Tsui; Jeffrey Wallin; Deepak Sampath; Alan Olivero
Bioorganic and Medicinal Chemistry Letters, ISSN: 14643405
Emily Hanan; Matt Baumgardner; Callie Bryan; Yuan Chen; Charles Eigenbrot; Peter Fan; Xiao-Hui Gu; Hank La; Shiva Malek; Hans Purkey; Gabriele Schaefer; Steve Schmidt; Steve Sideris; Ivana Yen; Christine Yu; Tim Heffron
ACS Medicinal Chemistry Letters, ISSN: 19485875
Callie Bryan; Dan Burdick; Bryan Chan; Yuan Chen; Saundra Clausen; Jenna Dotson; Charles Eigenbrot; Richard Elliott; Emily Hanan; Robert Heald; Philip Jackson; Hank La; Michael Lainchbury; Shiva Malek; Sam E. Mann; Hans Purkey; Gabriele Schaefer; Steve Schmidt; Eileen Seward; Steve Sideris; Shumei Wang; Ivana Yen; Christine Yu; Tim Heffron
ACS Symposium Series, ISSN: 19475918
Tim Heffron; Andrew McClory; Andy Stumpf
Journal of Medicinal Chemistry, ISSN: 15204804
Robert Heald; Krista Bowman; Callie Bryan; Dan Burdick; Bryan Chan; Emily Chan; Yuan Chen; Saundra Clausen; Belen Dominguez-Fernandez; Charles Eigenbrot; Richard Elliott; Emily Hanan; Philip Jackson; Jamie Knight; Hank La; Michael Lainchbury; Shiva Malek; Sam E. Mann; Mark Merchant; Kyle Mortara; Hans Purkey; Gabriele Schaefer; Stephen Schmidt; Eileen Seward; Steve Sideris; Lily Shao; Shumei Wang; Kuen Yeap; Ivana Yen; Christine Yu; Tim Heffron
Journal of Computer-Aided Molecular Design, ISSN: 15734951
Ignacio Aliagas; Alberto Gobbi; Tim Heffron; Man Ling Lee; Dan Ortwine; Mark Zak; Cyrus Khojasteh
Neuro-Oncology, ISSN: 15235866
Victor A. Levin; Peter J. Tonge; James M. Gallo; Marc R. Birtwistle; Arvin C. Dar; Antonio Iavarone; Patrick J. Paddison; Tim Heffron; William F. Elmquist; Jean E. Lachowicz; Ted W. Johnson; Forest M. White; Joohee Sul; Smith; Wang Shen; Jann N. Sarkaria; Ramakrishna Samala; Patrick Y. Wen; Donald A. Berry; Russell C. Petter
Journal of Medicinal Chemistry, ISSN: 15204804
Emily Hanan; Charles Eigenbrot; Callie Bryan; Dan Burdick; Bryan Chan; Yuan Chen; Jenna Dotson; Robert Heald; Philip Jackson; Hank La; Michael Lainchbury; Shiva Malek; Hans Purkey; Gabriele Schaefer; Steve Schmidt; Eileen M. Seward; Steve Sideris; Christine Tam; Shumei Wang; Siew Kuen Yeap; Ivana Yen; Peter Yin; Christine Yu; Inna Zilberleyb; Tim Heffron
Journal of Medicinal Chemistry, ISSN: 15204804
Tony Estrada; Bryan Chan; Charles Baker-Glenn; Alan Beresford; Dan Burdick; Mark Chambers; Huifen Chen; Sara Dominguez; Jenna Dotson; Jake Drummond; Mike Flagella; Reina Fuji; Andrew Gill; Jason Halladay; Seth Harris; Tim Heffron; Tracy Kleinheinz; Donna Lee; Claire Le Pichon; Xingrong Liu; Joe Lyssikatos; Andrew D. Medhurst; John Moffat; Kevin Nash; Kimberly Scearce-Levie; Zejuan Sheng; Daniel Shore; Susan Wong; Shuo Zhang; Xiaolin Zhang; Haitao Zhu; Zach Sweeney
Molecular Pharmaceutics, ISSN: 15438384
Gillian S. Smelick; Tim Heffron; Laura Chu; Brian Dean; David West; Scott L. Duvall; Bert Lum; Nageshwar Budha; Scott Holden; Leslie Z. Benet; Adam Frymoyer; Mark Dresser; Joseph Ware
Journal of Medicinal Chemistry, ISSN: 00222623
Chudi Ndubaku; Tim Heffron; Steven Staben; Matt Baumgardner; Nicole Blaquiere; Erin Bradley; Richard J. Bull; Steven Do; Jenna Dotson; Danette Dudley; Kyle Edgar; Lori Friedman; Rich Goldsmith; Robert Heald; Aleksandr Kolesnikov; Leslie Lee; Cris Lewis; Michelle Nannini; Jim Nonomiya; Jodie Pang; Steve Price; Wei Wei Prior; Laurent Salphati; Steve Sideris; Jeffrey Wallin; Lan Wang; Binqing Wei; Deepak Sampath; Alan Olivero
Bioorganic and Medicinal Chemistry Letters, ISSN: 0960894X
Steven Staben; Chudi Ndubaku; Nicole Blaquiere; Marcia Belvin; Richard J. Bull; Danette Dudley; Kyle Edgar; Daniel Gray; Robert Heald; Tim Heffron; Graham E. Jones; Mark Jones; Aleksandr Kolesnikov; Leslie Lee; John Lesnick; Cris Lewis; Jeremy Murray; Neville J. McLean; Jim Nonomiya; Alan Olivero; Rachel Ord; Jodie Pang; Stephen Price; Wei Wei Prior; Lionel Rouge; Laurent Salphati; Deepak Sampath; Jeffrey Wallin; Lan Wang; Binqing Wei; Christian Weismann; Ping Wu
Cancer Discovery, ISSN: 21598274
Ho-June Lee; Gabriele Schaefer; Tim Heffron; Lily Shao; Xiaofen Ye; Steve Sideris; Shiva Malek; Emily Chan; Mark Merchant; Hank La; Savita Ubhayakar; Bob Yauch; Valentina Pirazzoli; Katerina Politi; Jeffrey Settleman
Bioorganic and Medicinal Chemistry Letters, ISSN: 0960894X
Steven Staben; Nicole Blaquiere; Vickie Tsui; Aleksandr Kolesnikov; Steven Do; Erin Bradley; Jenna Dotson; Rich Goldsmith; Tim Heffron; John Lesnick; Cris Lewis; Jeremy Murray; Jim Nonomiya; Alan Olivero; Jodie Pang; Lionel Rouge; Laurent Salphati; Binqing Wei; Christian Wiesmann; Ping Wu
Journal of Medicinal Chemistry, ISSN: 00222623
Tony Estrada; Xingrong Liu; Charles Baker-Glenn; Alan Beresford; Dan Burdick; Mark Chambers; Bryan Chan; Huifen Chen; Xiao Ding; Antonio DiPasquale; Sara Dominguez; Jenna Dotson; Jake Drummond; Mike Flagella; Sean Flynn; Reina Fuji; Andrew Gill; Janet Gunzner-Toste; Seth Harris; Tim Heffron; Tracy Kleinheinz; Donna Lee; Claire Le Pichon; Joe Lyssikatos; Andrew D. Medhurst; John Moffat; Susmith Mukund; Kevin Nash; Kimberly Scearce-Levie; Zejuan Sheng; Daniel Shore; Thuy Tran; Naimisha Trivedi; Shumei Wang; Shuo Zhang; Xiaolin Zhang; Guiling Zhao; Haitao Zhu; Zach Sweeney
Clinical Cancer Research, ISSN: 10780432
Laurent Salphati; Tim Heffron; Bruno Alicke; Merry Nishimura; Kai Barck; Rick Carano; Jonathan Cheong; Kyle Edgar; Joan Greve; Samir Kharbanda; Hartmut Koeppen; Shari Lau; Leslie Lee; Jodie Pang; Emile Plise; Jenny L. Pokorny; Hani Bou-Reslan; Jann N. Sarkaria; Jeffrey Wallin; Xiaolin Zhang; Stephen Gould; Alan Olivero; Heidi Phillips
Journal of Medicinal Chemistry, ISSN: 00222623
Tim Heffron; Laurent Salphati; Bruno Alicke; Jonathan Cheong; Jenna Dotson; Kyle Edgar; Rich Goldsmith; Stephen Gould; Leslie Lee; John Lesnick; Cris Lewis; Chudi Ndubaku; Jim Nonomiya; Alan Olivero; Jodie Pang; Emile Plise; Steve Sideris; Sean Trapp; Jeffrey Wallin; Lan Wang; Xiaolin Zhang
Journal of Chemical Information and Modeling, ISSN: 15205142
Man Ling Lee; Ignacio Aliagas; Jenna Dotson; JW Feng; Alberto Gobbi; Tim Heffron
Journal of Medicinal Chemistry, ISSN: 00222623
Tim Heffron; Binqing Wei; Alan Olivero; Steven Staben; Vickie Tsui; Steven Do; Jenna Dotson; Adrian J. Folkes; Paul Goldsmith; Rich Goldsmith; Janet Gunzner-Toste; John Lesnick; Cris Lewis; Simon Mathieu; Jim Nonomiya; Stephen Shuttleworth; Dan Sutherlin; Nan Chi Wan; Shumei Wang; Christian Wiesmann; Bing-Yan Zhu
Journal of Medicinal Chemistry, ISSN: 00222623
Dan Sutherlin; Linda Bao; Megan Berry Swadell; Georgette Castanedo; Irina Chuckowree; Jenna Dotson; Adrian Folks; Lori Friedman; Rich Goldsmith; Janet Gunzner-Toste; Tim Heffron; John Lesnick; Cris Lewis; Simon Mathieu; Jeremy Murray; Jim Nonomiya; Jodie Pang; Neil Pegg; Wei Wei Prior; Lionel Rouge; Laurent Salphati; Deepak Sampath; Qingping Tian; Vickie Tsui; Nan Chi Wan; Shumei Wang; Binqing Wei; Christian Wiesmann; Ping Wu; Bing-Yan Zhu; Alan Olivero
Bioorganic and Medicinal Chemistry Letters, ISSN: 0960894X
Steven Staben; Mike Siu; Rich Goldsmith; Alan Olivero; Steven Do; Dan Burdick; Tim Heffron; Jenna Dotson; Dan Sutherlin; Bing-Yan Zhu; Vickie Tsui; Hoa Le; Leslie Lee; John Lesnick; Cris Lewis; Jeremy Murray; Jim Nonomiya; Jodie Pang; Wei Wei Prior; Laurent Salphati; Lionel Rouge; Deepak Sampath; Steve Sideris; Christian Wiesmann; Ping Wu
Bioorganic and Medicinal Chemistry Letters, ISSN: 0960894X
Steven Staben; Tim Heffron; Dan Sutherlin; Seema Bhat; Georgette Castanedo; Irina Chuckowree; Jenna Dotson; Adrian J. Folkes; Lori Friedman; Leslie Lee; John Lesnick; Cris Lewis; Jeremy Murray; Jim Nonomiya; Alan Olivero; Emile Plise; Jodie Pang; Wei Wei Prior; Laurent Salphati; Lionel Rouge; Deepak Sampath; Vickie Tsui; Nan Chi Wan; Shumei Wang; Christian Weismann; Ping Wu; Bing-Yan Zhu
Journal of Organic Chemistry, ISSN: 00223263
Tim Heffron; Graham L. Simpson; Estibaliz Merino; Timothy F. Jamison
Bioorganic and Medicinal Chemistry Letters, ISSN: 0960894X
Tim Heffron; Megan Berry Swadell; Georgette Castanedo; Christine Chang; Irina Chuckowree; Jenna Dotson; Adrian J. Folkes; Janet Gunzner-Toste; John Lesnick; Cris Lewis; Simon Mathieu; Jim Nonomiya; Alan Olivero; Jodie Pang; David Peterson; Laurent Salphati; Deepak Sampath; Steve Sideris; Dan Sutherlin; Vickie Tsui; Nan Chi Wan; Shumei Wang; Susan Wong; Bing-Yan Zhu
Journal of Medicinal Chemistry, ISSN: 00222623
Dan Sutherlin; Deepak Sampath; Megan Berry Swadell; Georgette Castanedo; Zhigang Chang; Irina Chuckowree; Jenna Dotson; Adrian J. Folkes; Lori Friedman; Rich Goldsmith; Tim Heffron; Leslie Lee; John Lesnick; Cris Lewis; Simon Mathieu; Jim Nonomiya; Alan Olivero; Jodie Pang; Wei Wei Prior; Laurent Salphati; Steve Sideris; Qingping Tian; Vickie Tsui; Nan Chi Wan; Shumei Wang; Christian Wiesmann; Susan Wong; Bing-Yan Zhu
Synlett, ISSN: 09365214
Tim Heffron; Timothy F. Jamison