Characterization of Tissue Distribution, Catabolism, and Elimination of an Anti-Staphylococcus aureus THIOMAB Antibody-Antibiotic Conjugate in Rats
Drug Metabolism and Disposition,
Hao Cai; Victor Yip; Violet Lee; Sylvia Wong; Ola Saad; Shuguang Ma; Nina Ljumanovic; S Cyrus Khojasteh; Amrita Kamath; Ben-Quan Shen
Systematic Variation of Pyrrolobenzodiazepine (PBD)-Dimer Payload Physicochemical Properties Impacts Efficacy and Tolerability of the Corresponding Antibody-Drug Conjugates
Journal of Medicinal Chemistry,
Leanna Staben; Jinhua Chen; Josefa Dela Cruz-Chuh; Geoff Del Rosario; Mary Ann Go; Jun Guo; S Cyrus Khojasteh; Kathy Kozak; Ginny Li; Carl Ng; Gail D. Lewis Phillips; Thomas Pillow; Rebecca K. Rowntree; John Wai; Binqing Wei; Keyang Xu; Zijin Xu; Shang-Fan Yu; Donglu Zhang; Peter Dragovich
Chemical Research in Toxicology, ISSN: 15205010
Chenghong Zhang; James Crawford; Matthew L. Landry; Huifen Chen; Jane Kenny; S Cyrus Khojasteh; Wendy Lee; Shuguang Ma; Wendy B. Young
Drug Metabolism and Disposition, ISSN: 1521009X 00909556
Haeyoung Zhang; Chris Wolford; Abdul Basit; Albert P. Li; Peter Fan; Bernard P. Murray; Ryan Takahashi; Cyrus Khojasteh; Bill J. Smith; Kenneth E. Thummel; Bhagwat Prasad
Xenobiotica, ISSN: 13665928 00498254
Wei Wang; Mulder Teresa; Jingwei Cai; Chenghong Zhang; Susan Wong; Zhengyin Yan; S Cyrus Khojasteh; Donglu Zhang
Carfilzomib Is Not an Appropriate Payload of Antibody-Drug Conjugates Due to Rapid Inactivation by Lysosomal Enzymes
Drug Metabolism and Disposition,
Yong Ma; Josefa Dela Cruz Chuh; S Cyrus Khojasteh; Peter Dragovich; Thomas Pillow; Donglu Zhang
Molecular Pharmaceutics, ISSN: 15438392 15438384
Zhonghua Pei; Chunjiao Chen; Jinhua Chen; Josefa Dela Cruz-Chuh; Reginald Delarosa; Yuzhong Deng; Aimee Fourie-O'Donohue; Isabel Figueroa; Jun Guo; Weiwei Jin; Cyrus Khojasteh; Kathy Kozak; Brandon Latifi; James Lee; Ginny Li; Eva Lin; Liling Liu; Jiawei Lu; Scott Martin; Carl Ng; Trung Nguyen; Rachana Ohri; Gail Phillips; Thomas Pillow; Rebecca K. Rowntree; Nicola Stagg; David Stokoe; Sheila Ulufatu; Vishal Verma; John Wai; Jing Wang; Keyang Xu; Zijin Xu; Hui Yao; Shang-Fan Yu; Donglu Zhang; Peter Dragovich
Drug Metabolism and Disposition, ISSN: 1521009X 00909556
Simone Schadt; Bojan Bister; Swapan K. Chowdhury; Christoph Funk; Marcel Hop; W. Griffith Humphreys; Fumihiko Igarashi; D James Alexander; Mark Kagan; Cyrus Khojasteh; Angus N. R Nedderman; Chandra Prakash; Frank Runge; Holger Scheible; Douglas K Spracklin; Piet Swart; Susanna Tse; Josh Yuan; R. Scott Obach
Molecular Cancer Therapeutics, ISSN: 15388514 15357163
Donglu Zhang; Shang-Fan Yu; Cyrus Khojasteh; Yong Ma; Thomas Pillow; Jack D. Sadowsky; Dian Su; Kathy Kozak; Keyang Xu; Andy Polson; Peter Dragovich; Marcel Hop
Bioconjugate Chemistry, ISSN: 15204812 10431802
Donglu Zhang; Hoa Le; Josefa Dela Cruz-Chuh; Sudheer Bobba; Jun Guo; Leanna Staben; Chenghong Zhang; Yong Ma; Kathy Kozak; Gail Phillips; Breanna S. Vollmar; Jack D. Sadowsky; Dick Vandlen; Binqing Wei; Dian Su; Peter Fan; Peter Dragovich; Cyrus Khojasteh; Marcel Hop; Thomas Pillow
British Journal of Clinical Pharmacology, ISSN: 13652125 03065251
Tore Bjerregaard Stage; Magnus Graff; Susan Wong; Louise Ladebo Rasmussen; Flemming Nielsen; Anton Pottegård; Kim Brøsen; Deanna L. Kroetz; Cyrus Khojasteh; Per Damkier
Minimal physiologically-based pharmacokinetic modeling of DSTA4637A, A novel THIOMAB™ antibody antibiotic conjugate against Staphylococcus aureus, in a mouse model
mAbs, ISSN: 19420862
Shun xin Wang-Lin; Chenguang Zhou; Amrita Kamath; Kyu Hong; Neelima Koppada; Ola Saad; Montse Carrasco-Triguero; Cyrus Khojasteh; Rong Deng
Glucuronides as Potential Anionic Substrates of Human Cytochrome P450 2C8 (CYP2C8)
Journal of Medicinal Chemistry, ISSN: 00222623
Yong Ma; Yue Fu; Cyrus Khojasteh; Deepak Dalvie; Donglu Zhang
CYP1A1-mediated intramolecular rearrangement of aminoazepane in GDC-0339
Drug Metabolism and Disposition, ISSN: 00909556
Ryan Takahashi; Gina Wang; Nathaniel Segraves; Jing Wang; Jae Chang; Cyrus Khojasteh; Shuguang Ma
Inhibitory effects of trapping agents of sulfur drug reactive intermediates against major human cytochrome P450 isoforms
International Journal of Molecular Sciences, ISSN: 16616596
Jasleen K. Sodhi; Erlie Delarosa; Jason Halladay; James Driscoll; Teresa Mulder; Patrick M. Dansette; Cyrus Khojasteh
Biotransformation and bioactivation reactions–2016 literature highlights
Drug Metabolism Reviews, ISSN: 03602532
Cyrus Khojasteh; Ivonne M. C. M. Rietjens; Deepak Dalvie; Grover Miller
Drug Metabolism and Disposition, ISSN: 1521009X
Ryan Takahashi; Jason Halladay; Mike Siu; Yuan Chen; Marcel Hop; Cyrus Khojasteh; Shuguang Ma
Drug Metabolism Letters, ISSN: 18723128
Ryan Takahashi; Cyrus Khojasteh; Matthew Wright; Marcel Hop; Shuguang Ma
Xenobiotica, ISSN: 13665928
Ryan Takahashi; Shuguang Ma; Qin Yue; Heasook Kim-Kang; Yijun Yi; Justin Ly; Jason Boggs; Alec Fettes; Andrew McClory; Yuzhong Deng; Marcel Hop; Cyrus Khojasteh; Edna Choo
Drug Metabolism and Disposition, ISSN: 1521009X
Yong Ma; Cyrus Khojasteh; Marcel Hop; Hans Erickson; Andy Polson; Thomas Pillow; Shang-Fan Yu; Hong Wang; Peter Dragovich; Donglu Zhang
ACS Medicinal Chemistry Letters, ISSN: 19485875
Donglu Zhang; Thomas Pillow; Yong Ma; Josefa Dela Cruz-Chuh; Kathy Kozak; Jack Sadowsky; Gail Phillips; Jun Guo; Martine Darwish; Peter Fan; Jingtian Chen; Changrong He; Tao Wang; Hui Yao; Zijin Xu; Jinhua Chen; John Wai; Zhonghua Pei; Marcel Hop; Cyrus Khojasteh; Peter Dragovich
Drug Metabolism and Disposition, ISSN: 1521009X
Donglu Zhang; Shang-Fan Yu; Yong Ma; Keyang Xu; Peter Dragovich; Thomas Pillow; Luna Liu; Geoff Del Rosario; Jintang He; Zhonghua Pei; Jack Sadowsky; Hans Erickson; Marcel Hop; Cyrus Khojasteh
Drug Metabolism and Disposition, ISSN: 1521009X
Peter Fan; Donglu Zhang; Jason Halladay; James Driscoll; Cyrus Khojasteh
Drug Metabolism Letters, ISSN: 18723128
Hoa Le; Peter Fan; Susan Wong; Shuguang Ma; James Driscoll; Marcel Hop; Cyrus Khojasteh
Drug Metabolism Letters, ISSN: 18723128
Peter Fan; Jacob Chen; Allan Jaochico; Hank La; Ning Liu; Teresa Mulder; Robert T. Cass; Matthew Durk; Kirsten Messick; Nicole Valle; Shannon Liu; Wendy Lee; James Crawford; Joachim Rudolph; Lesley Murray; Cyrus Khojasteh; Matthew Wright
Pharmaceutical Research, ISSN: 1573904X
Jialin Mao; Suzanne Brown; Cyrus Khojasteh; Yuan Chen; Marcel Hop; Jane Kenny
Drug Metabolism and Disposition, ISSN: 1521009X
Ryan Takahashi; Edna Choo; Shuguang Ma; Susan Wong; Jason Halladay; Yuzhong Deng; Isabelle Rooney; Mary Gates; Marcel Hop; Cyrus Khojasteh; Mark Dresser; Luna Musib
Drug Metabolism and Disposition, ISSN: 1521009X
Ryan Takahashi; Shuguang Ma; Sarah Robinson; Qin Yue; Edna Choo; Cyrus Khojasteh
Drug Metabolism and Disposition, ISSN: 1521009X
Jasleen K. Sodhi; Susan Wong; Don Kirkpatrick; Lichuan Liu; Cyrus Khojasteh; Marcel Hop; John T. Barr; Jeffrey P. Jones; Jason Halladay
European Journal of Drug Metabolism and Pharmacokinetics, ISSN: 21070180
Ryan Takahashi; Shuguang Ma; Qin Yue; Heasook Kim-Kang; Yijun Yi; Joe Lyssikatos; Kelly Regal; Kevin W. Hunt; Nicholas C. Kallan; Mike Siu; Marcel Hop; Xingrong Liu; Cyrus Khojasteh
Journal of Computer-Aided Molecular Design, ISSN: 15734951
Ignacio Aliagas; Alberto Gobbi; Tim Heffron; Man Ling Lee; Dan Ortwine; Mark Zak; Cyrus Khojasteh
Drug Metabolism Reviews, ISSN: 10979883
Perry Gordon; Cyrus Khojasteh
Bioanalysis, ISSN: 17576199
Ola Saad; Ben-Quan Shen; Keyang Xu; Cyrus Khojasteh; Sandhya Girish; Surinder Kaur
Drug Metabolism Letters, ISSN: 18723128
Ben-Quan Shen; Daniela Yadav; Qin Yue; Ola Saad; Jack (Jay) Tibbitts; Cyrus Khojasteh; Sandhya Girish
Drug Metabolism and Disposition, ISSN: 00909556
Cyrus Khojasteh; Qin Yue; Shuguang Ma; Georgette Castanedo; Jacob Chen; Joe Lyssikatos; Teresa Mulder; Ryan Takahashi; Justin Ly; Kirsten Messick; Wei Jia; Lichuan Liu; Marcel Hop; Harvey Wong
Drug Metabolism and Disposition, ISSN: 1521009X 00909556
Ryan Takahashi; Shuguang Ma; Alan Deese; Qin Yue; Heasook Kim-Kang; Yijun Yi; Mike Siu; Kevin W. Hunt; Nicholas C. Kallan; Marcel Hop; Xingrong Liu; Cyrus Khojasteh
Toxicology Research, ISSN: 20454538
Chenghong Zhang; Shuguang Ma; Erlie Delarosa; Suzanne Brown; Jasleen K. Sodhi; Vivek Musinipally; Patricia Chang; Rama Pai; Jason Halladay; Misner; Jane Kenny; Marcel Hop; Cyrus Khojasteh
Drug Metabolism and Disposition, ISSN: 1521009X
Suzanne Tay; Hoa Le; Kevin Ford; Sidney D. Nelson; Cyrus Khojasteh; Peter M. Rademacher
Future Medicinal Chemistry, ISSN: 17568927
Peter Fan; Yang Song; Leo Berezhkovskiy; Jonathan Cheong; Emile Plise; Cyrus Khojasteh
Drug Metabolism and Disposition, ISSN: 1521009X
Jasleen K. Sodhi; Kevin Ford; Sophie Aurangabadwala; Susan Wong; Marcel Hop; Cyrus Khojasteh; Jason Halladay
Clinical Pharmacology and Therapeutics, ISSN: 00099236
Markova; Teresa De Marco; Bendjilali; Kobashigawa; Mefford; Jasleen K. Sodhi; Le; Zhang; Jason Halladay; Rettie; Cyrus Khojasteh; McGlothlin; Wu; Hsueh; Witte; Schwartz; Deanna L. Kroetz
Bioorganic and Medicinal Chemistry Letters, ISSN: 0960894X
Mike Siu; Rich Pastor; Wendy Liu; Kathy Barrett; Megan Berry Swadell; Wade Blair; Christine Chang; Jacob Chen; Charles Eigenbrot; Nico Ghilardi; Paul Gibbons; Haiying He; Christopher A. Hurley; Jane Kenny; Cyrus Khojasteh; Hoa Le; Leslie Lee; Joe Lyssikatos; Steven Magnuson; Rebecca Pulk; Vickie Tsui; Mark Ultsch; Yisong Xiao; Bing-Yan Zhu; Deepak Sampath
Xenobiotica, ISSN: 00498254
Hoa Le; Kevin Ford; Cyrus Khojasteh; Peter Fan
Drug Metabolism and Disposition, ISSN: 00909556
Qin Yue; Teresa Mulder; Patrick Rudewicz; Eric G. Solon; Nageshwar Budha; Joseph Ware; Joe Lyssikatos; Marcel Hop; Harvey Wong; Cyrus Khojasteh
Drug Metabolism Letters, ISSN: 18723128
Sophie Aurangabadwala; Suzanne Brown; Daniel Tran; Leslie Wang; Erlie Delarosa; Cyrus Khojasteh; Jason Halladay; Jane Kenny
Chemical Research in Toxicology, ISSN: 0893228X
Cyrus Khojasteh; Dylan Hartley; Kevin Ford; Hirdesh Uppal; Shimako Oishi; Sidney D. Nelson
Current Drug Metabolism, ISSN: 13892002
Ben-Quan Shen; Daniela Yadav; Ola Saad; Qin Yue; Cinthia Pastuskovas; Cyrus Khojasteh; Jack (Jay) Tibbitts; Surinder Kaur; Bei Wang; Wayne Chu; Patricia M. LoRusso; Sandhya Girish
Journal of Pharmacological and Toxicological Methods, ISSN: 10568719
Jason Halladay; Susan Wong; Cyrus Khojasteh; Susan Grepper
Pharmaceutical Research, ISSN: 07248741
Jane Kenny; Sophie Aurangabadwala; Chenghong Zhang; Suzanne Brown; Carol Collins; Aleksandra Galetin; Cyrus Khojasteh
Combinatorial Chemistry and High Throughput Screening, ISSN: 13862073
Young Shin; Hoa Le; Cyrus Khojasteh; Marcel Hop
Chemical Research in Toxicology, ISSN: 0893228X
Chenghong Zhang; Jane Kenny; Hoa Le; Alan Deese; Kevin Ford; Luke K. Lightning; Peter Fan; James Driscoll; Jason Halladay; Marcel Hop; Cyrus Khojasteh
Drug Metabolism and Disposition, ISSN: 00909556
Lichuan Liu; Jason Halladay; Young Shin; Susan Wong; Melis Coraggio; Hank La; Matt Baumgardner; Hoa Le; Sashi Gopaul; Jason Boggs; Peter Kuebler; John Davis; Charlene Liao; Joe Lubach; Alan Deese; Greg Sowell; Kevin S. Currie; Wendy Young; Cyrus Khojasteh; Marcel Hop; Harvey Wong
Drug Metabolism Letters, ISSN: 18723128
Jason Halladay; Erlie Delarosa; Daniel Tran; Leslie Wang; Susan Wong; Cyrus Khojasteh
Drug Metabolism and Disposition, ISSN: 00909556
Qin Yue; John Chen; Teresa Mulder; Alan Deese; Ryan Takahashi; Patrick Rudewicz; Mark Reynolds; Eric G. Solon; Marcel Hop; Harvey Wong; Cyrus Khojasteh
European Journal of Drug Metabolism and Pharmacokinetics, ISSN: 03787966
Cyrus Khojasteh; Saileta Prabhu; Jane Kenny; Jason Halladay; Anthony Y. H. Lu
Chemical Research in Toxicology, ISSN: 0893228X
Cyrus Khojasteh; Shimako Oishi; Sidney D. Nelson
Bioorganic and Medicinal Chemistry Letters, ISSN: 0960894X
Georgette Castanedo; Shumei Wang; Kirk Robarge; Beth Blackwood; Dan Burdick; Christine Chang; Peter Dijkgraaf; Stephen Gould; Janet Gunzner-Toste; Oivin Guichert; Jason Halladay; Cyrus Khojasteh; Leslie Lee; James Marsters; Lesley Murray; David Peterson; Emile Plise; Laurent Salphati; Frederic De Sauvage; Susan Wong; Dan Sutherlin
Chemical Research in Toxicology, ISSN: 0893228X
James Driscoll; Ignacio Aliagas; Jennifer Harris; Jason Halladay; Sheerin Latham; Alan Deese; Nathaniel Segraves; Cyrus Khojasteh
Bioorganic and Medicinal Chemistry Letters, ISSN: 0960894X
Kirk Robarge; Shirley A. Brunton; Georgette Castanedo; Yong Cui; Michael Dina; Rich Goldsmith; Stephen Gould; Oivin Guichert; Janet Gunzner-Toste; Jason Halladay; Wei Jia; Cyrus Khojasteh; Michael Koehler; Karen Kotkow; Hank La; Rebecca Lyn K. LaLonde; Kevin Lau; Leslie Lee; Derek Marshall; James Marsters; Lesley Murray; Changgeng Qian; Lee L. Rubin; Laurent Salphati; Mark Stanley; John H.A. Stibbard; Dan Sutherlin; Savita Ubhayakar; Shumei Wang; Susan Wong; Minli Xie
Drug Metabolism and Disposition, ISSN: 1521009X
Harvey Wong; Peter Theil; Yong Cui; James Marsters; Cyrus Khojasteh; Laurent Vernillet; Hank La; Xiling Song; Hong Wang; Eric Morinello; Yuzhong Deng; Marcel Hop
Xenobiotica, ISSN: 00498254
Harvey Wong; Jian Chen; Bilin Chou; Jason Halladay; Jane Kenny; Hank La; James Marsters; Emile Plise; Patrick Rudewicz; Kirk Robarge; Young Shin; Susan Wong; Chenghong Zhang; Cyrus Khojasteh
Bioorganic and Medicinal Chemistry Letters, ISSN: 0960894X
Kirk Robarge; Shirley A. Brunton; Georgette Castanedo; Yong Cui; Michael Dina; Rich Goldsmith; Stephen Gould; Oivin Guichert; Janet Gunzner-Toste; Jason Halladay; Wei Jia; Cyrus Khojasteh; Michael Koehler; Karen Kotkow; Hank La; Rebecca Lyn K. LaLonde; Kevin Lau; Leslie Lee; Derek Marshall; James Marsters; Lesley Murray; Changgeng Qian; Lee L. Rubin; Laurent Salphati; Mark Stanley; John H.A. Stibbard; Dan Sutherlin; Savita Ubhayakar; Shumei Wang; Susan Wong; Minli Xie
Journal of Pharmaceutical Sciences, ISSN: 00223549
Leo Berezhkovskiy; Cyrus Khojasteh; Jason Halladay; Marcel Hop
Drug Metabolism Letters, ISSN: 18723128
Chenghong Zhang; Susan Wong; Erlie Delarosa; Jane Kenny; Jason S. Hallday; Marcel Hop; Cyrus Khojasteh
Xenobiotica, ISSN: 00498254
Cyrus Khojasteh; Douglas Leipold; Lai; Hank La; Matt Baumgardner; Desino; Olafur S. Gudmundsson; Duane Bloedow; Sarah C. Bodary; Mark Reynolds; Thomas R. Gadek; Sara Kenkare-Mitra
Drug Metabolism and Disposition, ISSN: 00909556
Chandra Prakash; John O'Donnell; Cyrus Khojasteh
Drug Metabolism Letters, ISSN: 18723128
Jason Halladay; Susan Wong; Sharmin M Jaffer; Achintya Sinhababu; Cyrus Khojasteh
Journal of Chromatography B: Analytical Technologies in the Biomedical and Life Sciences, ISSN: 15700232
Frances Y. Lai; Cyrus Khojasteh
Xenobiotica, ISSN: 00498254
Cyrus Khojasteh; Rossulek; Fouda; Chandra Prakash
Chemical Research in Toxicology, ISSN: 0893228X
Deepak Dalvie; Amit S. Kalgutkar; Cyrus Khojasteh; R. Scott Obach; John O'Donnell