Scientific Reports, ISSN: 20452322
Rebecca M. Reese; Michelle Dourado; Keith Anderson; Soren Warming; Kimberly L. Stark; Alessia Balestrini; Eric Suto; Wyne Lee; Lorena Riol Blanco; Shannon Shields; David Hackos
Cell Reports, ISSN: 22111247
Jesse E. Hanson; Keran Ma; Justin Elstrott; Martin Weber; Sandrine Saillet; Abdullah S. Khan; Jeffrey Simms; Benjamin Liu; Thomas A. Kim; Gui-Qiu Yu; Yelin Chen; Tzu-Ming Wang; Zhiyu Jiang; Bianca Liederer; Gauri Deshmukh; Hilda Solanoy; Connie Chan; Ben Sellers; Matthew Volgraf; Jacob Schwarz; David Hackos; Robby Weimer; Morgan Sheng; T. Michael Gill; Kimberly Scearce-Levie; Jorge J. Palop
A Non-covalent Ligand Reveals Biased Agonism of the TRPA1 Ion Channel
Neuron, ISSN: 08966273
Chang Liu; Rebecca M. Reese; Simon Vu; Lionel Rouge; Shannon Shields; Satoko Kakiuchi-Kiyota; Huifen Chen; Kevin Johnson; Yu Patrick Shi; Tania Chernov-Rogan; Demi Maria Zabala Greiner; Pawan Bir Kohli; David Hackos; Bobby Brillantes; Christine Tam; Tianbo Li; Jianyong Wang; Brian Safina; Steven Magnuson; Matthew Volgraf; Jian Payandeh; Jie Zheng; Alexis Rohou; Jun Chen
Proceedings of the National Academy of Sciences of the United States of America, ISSN: 10916490 00278424
Tania Chernov-Rogan; Eleonora Gianti; Chang Liu; Elisia Villemure; Andrew P. Cridland; Xiaoyu Hu; Elisa Ballini; Wienke Lange; Heike Deisemann; Tianbo Li; Stuart I. Ward; David Hackos; Steven Magnuson; Brian Safina; Michael L. Klein; Matthew Volgraf; Vincenzo Carnevale; Jun Chen
Science, ISSN: 10959203 00368075
Thomas Clairfeuille; Alexander Cloake; Daniel T. Infield; José P. Llongueras; Christopher P. Arthur; Zhong Rong Li; Yuwen Jian; Marie-France Martin-Eauclaire; Pierre E. Bougis; Claudio Ciferri; Christopher A. Ahern; Frank Bosmans; David Hackos; Alexis Rohou; Jian Payandeh
Structural Basis of Nav1.7 Inhibition by a Gating-Modifier Spider Toxin
Cell, ISSN: 00928674
Hui Xu; Tianbo Li; Alexis Rohou; Christopher P. Arthur; Foteini Tzakoniati; Evera Wong; Alberto Estevez; Christine Kugel; Yvonne Franke; Jun Chen; Claudio Ciferri; David Hackos; Chris Koth; Jian Payandeh
Journal of Medicinal Chemistry, ISSN: 15204804 00222623
Steven J. McKerrall; Teresa Nguyen; Kwong Wah Lai; Philippe Bergeron; Lunbin Deng; Antonio DiPasquale; Jae Chang; Jun Chen; Tania Chernov-Rogan; David Hackos; Jonathan M. Maher; Dan Ortwine; Jodie Pang; Jian Payandeh; Will Proctor; Shannon Shields; Jennifer Vogt; Pengfei Ji; Wenfeng Liu; Elisa Ballini; Lilia Schumann; Glauco Tarozzo; Girish Bankar; Sultan Chowdhury; Abid Hasan; Johnson; Kuldip Khakh; Sophia Lin; Charles J. Cohen; Christoph Dehnhardt; Brian Safina; Dan Sutherlin
Clinical Drug Investigation, ISSN: 11791918 11732563
Michael E. Rothenberg; Tagen; Jae H. Chang; Janel Boyce-Rustay; Michel Friesenhahn; David Hackos; Avis Hains; Dan Sutherlin; Michael Ward; William Cho
Safety, Tolerability, and Pharmacokinetics of GDC-0276, a Novel NaV1.7 Inhibitor, in a First-in-Human, Single- and Multiple-Dose Study in Healthy Volunteers
Clinical Drug Investigation, ISSN: 11732563
Michael E. Rothenberg; Tagen; Jae H. Chang; Janel Boyce-Rustay; Michel Friesenhahn; David Hackos; Avis Hains; Dan Sutherlin; Michael Ward; William Cho
Insensitivity to Pain upon Adult-Onset Deletion of Nav1.7 or Its Blockade with Selective Inhibitors
Journal of Neuroscience,
Shannon Shields; Lunbin Deng; Rebecca M. Reese; Michelle Dourado; Janet Tao; Oded Foreman; Jae H. Chang; David Hackos
Cell Reports, ISSN: 22111247
Girish Bankar; Samuel J. Goodchild; Sarah Howard; Karen Nelkenbrecher; Matthew Waldbrook; Michelle Dourado; Noah Shuart; Sophia Lin; Clint Young; Zhiwei Xie; Kuldip Khakh; Elaine Chang; Luis E. Sojo; Andrea Lindgren; Sultan Chowdhury; Shannon M. Decker; Michael Grimwood; Jean-Christophe Andrez; Christoph Dehnhardt; Jodie Pang; Jae H. Chang; Brian Safina; Dan Sutherlin; James P. Johnson; David Hackos; C. Lee Robinette; Charles J. Cohen
Journal of Medicinal Chemistry, ISSN: 15204804 00222623
Thilo Focken; Sultan Chowdhury; Alla Zenova; Michael Grimwood; Christine Chabot; Tao Sheng; Ivan Hemeon; Shannon M. Decker; Michael Wilson; Paul Bichler; Qi Jia; Shaoyi Sun; Clint Young; Sophia Lin; Samuel J. Goodchild; Noah Shuart; Elaine Chang; Zhiwei Xie; Bowen Li; Kuldip Khakh; Girish Bankar; Matthew Waldbrook; Rainbow Kwan; Karen Nelkenbrecher; Parisa Karimi Tari; Navjot Chahal; Luis E. Sojo; C. Lee Robinette; Andrew D. White; Chien-An Chen; Yi Zhang; Jodie Pang; Jae Chang; David Hackos; Johnson; Charles J. Cohen; Dan Ortwine; Dan Sutherlin; Christoph Dehnhardt; Brian Safina
Journal of Medicinal Chemistry, ISSN: 15204804 00222623
Huifen Chen; Matthew Volgraf; Steven Do; Aleksandr Kolesnikov; Daniel Shore; Vishal Verma; Elisia Villemure; Lan Wang; Yong Chen; Baihua Hu; Aijun Lu; Guosheng Wu; Xiaofeng Xu; Po-Wai Yuen; Yamin Zhang; Shawn D. Erickson; Martin Dahl; Christine Brotherton-Pleiss; Suzanne Brown; Justin Ly; Lesley Murray; Jun Chen; Desiree Amm; Wienke Lange; David Hackos; Rebecca M. Reese; Shannon Shields; Joe Lyssikatos; Brian Safina; Tony Estrada
Mechanism-specific assay design facilitates the discovery of Nav1.7-selective inhibitors
Proceedings of the National Academy of Sciences of the United States of America, ISSN: 00278424
Tania Chernov-Rogan; Tianbo Li; Gang Lu; Henry Verschoof; Kuldip Khakh; Steven W Jones; Maureen Beresini; Chang Liu; Dan Ortwine; Steven J. McKerrall; David Hackos; Dan Sutherlin; Charles J. Cohen; Jun Chen
Journal of Medicinal Chemistry, ISSN: 15204804 00222623
Shaoyi Sun; Qi Jia; Alla Zenova; Michael S. Wilson; Sultan Chowdhury; Thilo Focken; Jun Li; Shannon M. Decker; Michael Grimwood; Jean-Christophe Andrez; Ivan Hemeon; Tao Sheng; Chien-An Chen; Andrew D. White; David Hackos; Lunbin Deng; Girish Bankar; Kuldip Khakh; Elaine Chang; Rainbow Kwan; Sophia Lin; Karen Nelkenbrecher; Ben Sellers; Antonio DiPasquale; Jae H. Chang; Jodie Pang; Luis E. Sojo; Andrea Lindgren; Matthew Waldbrook; Zhiwei Xie; Clint Young; James P. Johnson; C. Lee Robinette; Charles J. Cohen; Brian Safina; Dan Sutherlin; Dan Ortwine; Christoph Dehnhardt
Handbook of Experimental Pharmacology, ISSN: 18650325 01712004
Jian Payandeh; David Hackos
Neuropharmacology, ISSN: 18737064
Tzu-Ming Wang; Brandon M. Brown; Lunbin Deng; Ben Sellers; Patrick Lupardus; Heidi Ackerly Wallweber; Amy Gustafson; Evera Wong; Matthew Volgraf; Jacob Schwarz; David Hackos; Jesse Hanson
Scientific Reports, ISSN: 20452322
Anton V. Sinitskiy; Nathaniel H. Stanley; David Hackos; Jesse Hanson; Ben Sellers; Vijay S. Pande
Nature Communications, ISSN: 20411723
Eugene Chiang; Tianbo Li; Surinder Jeet; Peng; Juan Zhang; Wyne Lee; Jason DeVoss; Patrick Caplazi; Jun Chen; Soren Warming; David Hackos; Susmith Mukund; Chris Koth; Jane Grogan
ACS Medicinal Chemistry Letters, ISSN: 19485875
Elisia Villemure; Matthew Volgraf; Yu Jiang; Guosheng Wu; Cuong Ly; Po-Wai Yuen; Aijun Lu; Xifeng Luo; Mingcui Liu; Shun Zhang; Patrick Lupardus; Heidi Ackerly Wallweber; Bianca Liederer; Gauri Deshmukh; Emile Plise; Suzanne Brown; Tzu-Ming Wang; Jesse Hanson; David Hackos; Kimberly Scearce-Levie; Jacob Schwarz; Ben Sellers
Journal of Medicinal Chemistry, ISSN: 15204804
Matthew Volgraf; Ben Sellers; Yu Jiang; Guosheng Wu; Cuong Ly; Elisia Villemure; Rich Pastor; Po-Wai Yuen; Aijun Lu; Xifeng Luo; Mingcui Liu; Shun Zhang; Liang Sun; Yuhong Fu; Patrick Lupardus; Heidi Ackerly Wallweber; Bianca Liederer; Gauri Deshmukh; Emile Plise; Suzanne Brown; Paul Reynen; James Herrington; Amy Gustafson; Yichin Liu; Akim Dirksen; Matthias G. A. Dietz; Yanzhou Liu; Tzu-Ming Wang; Jesse Hanson; David Hackos; Kimberly Scearce-Levie; Jacob Schwarz
Neuron, ISSN: 10974199
David Hackos; Patrick Lupardus; Teddy Grand; Yelin Chen; Tzu-Ming Wang; Paul Reynen; Amy Gustafson; Heidi Ackerly Wallweber; Matthew Volgraf; Ben Sellers; Jacob Schwarz; Pierre Paoletti; Morgan Sheng; Qiang Zhou; Jesse Hanson
Bioorganic and Medicinal Chemistry Letters, ISSN: 14643405
Vishal Verma; Daniel Shore; Huifen Chen; Jun Chen; Steven Do; David Hackos; Aleksandr Kolesnikov; Joe Lyssikatos; Suzanne Brown; Lan Wang; Tony Estrada
Science, ISSN: 10959203
Shivani Ahuja; Susmith Mukund; Lunbin Deng; Kuldip Khakh; Elaine Chang; Hoangdung Ho; Stephanie Shriver; Clint Young; Sophia Lin; Johnson; Ping Wu; Jun Li; Mary Coons; Christine Tam; Bobby Brillantes; Honorio Sampang; Kyle Mortara; Krista Bowman; Kevin Clark; Alberto Estevez; Zhiwei Xie; Henry Verschoof; Michael Grimwood; Christoph Dehnhardt; Jean-Christophe Andrez; Thilo Focken; Dan Sutherlin; Brian Safina; Melissa Starovasnik; Dan Ortwine; Yvonne Franke; Charles J. Cohen; David Hackos; Chris Koth; Jian Payandeh
Naunyn-Schmiedeberg's Archives of Pharmacology, ISSN: 14321912
Jun Chen; David Hackos
PLoS ONE, ISSN: 19326203
Michelle Dourado; Evera Wong; David Hackos
Journal of Neuroscience, ISSN: 02706474
Jesse Hanson; Lunbin Deng; David Hackos; Shih-Ching Lo; Ben Lauffer; Pascal Steiner; Qiang Zhou
Journal of Immunology, ISSN: 00221767
Yan Qu; Shahram Misaghi; Kim Newton; Laurie Appling; Salina Louie; Jim Cupp; George R. Dubyak; David Hackos; Vishva Dixit
British Journal of Pharmacology, ISSN: 14765381
Joel R. Gever; Rothschild Soto; Robert A. Henningsen; Renee S. Martin; David Hackos; Sandip Panicker; Werner Rubas; Ian B. Oglesby; Michael P. Dillon; Marcos E. Milla; Geoffrey Burnstock; Anthony P. D. W. Ford